SCHEMBL7708256

SCHEMBL7708256

CCCCCCNc1nc(NC[C@H](O)c2ccccc2)c2ncn(C(C)C)c2n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 13/20 0.70
CDK5 Q00535 6/20 0.70
CDK2 P24941 10/20 0.60
CCNB1 P14635 6/20 0.60
CCNB2 O95067 4/20 0.60
CCNB3 Q8WWL7 4/20 0.60
TDP1 Q9NUW8 2/20 0.60
CSNK1D P48730 1/20 0.57
CLK2 P49760 1/20 0.57
DYRK1A Q13627 1/20 0.57
HIPK4 Q8NE63 1/20 0.57
SRPK1 Q96SB4 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
CCNE1 P24864 5/20 0.56
CCNE2 O96020 3/20 0.56
CCNA2 P20248 3/20 0.56
CCNA1 P78396 3/20 0.56
KDM4E B2RXH2 1/20 0.56
NPC1 O15118 1/20 0.56
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7707862 0.88 CDK1 (0.75) CDK1CDK5CDK2CCNB1CCNB2
SCHEMBL6016445 0.84 CDK1 (0.66) CDK1CDK5CDK2CCNB1CCNB2
SCHEMBL6016435 0.84 CDK1 (0.66) CDK1CDK5CDK2CCNB1CCNB2
SCHEMBL7711075 0.80 CDK1 (0.69) CDK1CDK5CDK2CCNB1TDP1
SCHEMBL7113555 0.78 CDK1 (0.92) CDK1CDK5CDK2CCNB1CCNB2
SCHEMBL7112489 0.77 CDK1 (0.94) CDK1CDK5CDK2CCNB1CCNB2
SCHEMBL31069517 0.76 TDP1 (0.87) CDK1CDK5CDK2CCNB1CCNB2
Bohemine SCHEMBL1443403 0.75 CDK1 (1.00) CDK1CDK5CDK2CCNB1CCNB2
SCHEMBL7707886 0.74 CDK1 (0.60) CDK1CDK5CDK2CCNB1CSNK1D
SCHEMBL24669662 0.73 TDP1 (0.81) CDK1CDK5CDK2CCNB1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244668-A1 PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 2002-10-02 EP disclosed
WO-2001049688-A1 PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 2001-07-12 WO disclosed