SCHEMBL7708301

SCHEMBL7708301

CC(c1ccc(O)c(O)c1)c1nc(N)nc2c1ncn2C(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 9/20 0.53
CCNE1 P24864 7/20 0.53
CDK1 P06493 5/20 0.53
CCNB1 P14635 3/20 0.53
PRKACA P17612 1/20 0.44
CCNA2 P20248 1/20 0.44
PRKACG P22612 1/20 0.44
PRKACB P22694 1/20 0.44
MAPK3 P27361 1/20 0.44
MAPK1 P28482 1/20 0.44
CCNA1 P78396 1/20 0.44
CCNE2 O96020 2/20 0.41
ADORA2A P29274 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
HDAC8 Q9BY41 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
PI4KA P42356 1/20 0.39
PI4K2B Q8TCG2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21540017 0.74 CDK1 (0.71) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL7708273 0.72 TDP1 (0.37) MAPK1ADORA2AADORA2BADORA1PI4KA
SCHEMBL6527244 0.71 CDK2 (0.57) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL756644 0.71 CDK1 (1.00) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL29611365 0.71 CDK1 (1.00) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL16080845 0.70 CDK2 (0.73) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL23641811 0.68 CDK1 (0.71) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL756290 0.68 CDK2 (0.71) CDK2CCNE1CDK1CCNB1PRKACA
SCHEMBL6016359 0.68 CCNB2 (0.54) CDK2CCNE1CDK1CCNB1CCNA2
SCHEMBL12451372 0.66 CDK1 (0.67) CDK2CCNE1CDK1CCNB1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244668-A1 PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 2002-10-02 EP claimed
WO-2001049688-A1 PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND USE THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 2001-07-12 WO claimed