SCHEMBL7708919

SCHEMBL7708919

COc1ccc(CNc2cc(N)n3nc(-c4ccco4)nc3c2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.56
ADORA1 P30542 9/20 0.56
ADORA3 P0DMS8 8/20 0.56
ADORA2B P29275 3/20 0.54
MAPT P10636 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703121 0.89 ADORA2A (0.62) ADORA2AADORA1ADORA3ADORA2BMAPT
SCHEMBL7431721 0.86 ADORA2A (0.56) ADORA2AADORA1ADORA3ADORA2BMAPT
SCHEMBL7703042 0.83 ADORA2A (0.52) ADORA2AMAPT
SCHEMBL7708996 0.83 ADORA3 (0.51) ADORA2AADORA1ADORA3ADORA2BMAPT
SCHEMBL6047269 0.81 ADORA2A (0.63) ADORA2AADORA1ADORA3ADORA2BMAPT
SCHEMBL6047324 0.80 ADORA2A (0.61) ADORA2AADORA1ADORA3ADORA2BMAPT
SCHEMBL6047265 0.80 ADORA2A (0.61) ADORA2AADORA1ADORA3ADORA2BMAPT
Hydrochloric Acid SCHEMBL6047292 0.80 ADORA2A (0.61) ADORA2AADORA1ADORA3
SCHEMBL7478262 0.79 ADORA2A (0.56) ADORA2AMAPT
SCHEMBL6047307 0.79 ADORA2A (0.61) ADORA2AADORA1ADORA3ADORA2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed