SCHEMBL7709254

SCHEMBL7709254

CC(C)(C)[Si](C)(C)Oc1ccccc1[C@H]1CC[C@@H](CO)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.40
ADRA2A P08913 5/20 0.40
SLC6A2 P23975 3/20 0.40
SLC6A4 P31645 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
ADRA1A P35348 2/20 0.40
CYP2C9 P11712 2/20 0.40
CHRM1 P11229 2/20 0.40
USP2 O75604 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
PTGS1 P23219 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
KCNH2 Q12809 1/20 0.40
HTR2C P28335 3/20 0.39
SSTR4 P31391 3/20 0.38
SSTR1 P30872 2/20 0.38
ADRA2B P18089 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6433400 0.84 CA12 (0.36) CYP2D6CYP2C9ESR1CYP3A4ESR2
SCHEMBL6433023 0.84 CA12 (0.36) CYP2D6CYP2C9ESR1CYP3A4ESR2
SCHEMBL6433716 0.84 CA12 (0.36) CYP2D6CYP2C9ESR1CYP3A4ESR2
SCHEMBL7701150 0.82 HTR2C (0.39) HTR1AADRA2ASLC6A2SLC6A4CYP1A2
SCHEMBL7137900 0.78 HTR2C (0.38) HTR1AADRA2ASLC6A2SLC6A4CYP1A2
SCHEMBL7706184 0.75 HCRTR2 (0.36) HTR1AADRA2ASLC6A2SLC6A4CYP1A2
SCHEMBL20524226 0.75 ESR2 (0.51) CYP2D6CYP2C9ESR1CYP3A4ESR2
SCHEMBL8705847 0.75 CNR2 (0.42) HTR1AADRA2ASLC6A2SLC6A4CYP1A2
SCHEMBL7213445 0.73 MAPT (0.44) CYP1A2CYP3A4LMNA
SCHEMBL18244622 0.71 ESR2 (0.56) CYP2D6CYP2C9ESR1CYP3A4ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165495-A1 RESORCINOL DERIVATIVES PFIZER INC. (US) 2002-01-02 EP disclosed
WO-2000056702-A1 RESORCINOL DERIVATIVES PFIZER INC. (US) 2000-09-28 WO disclosed