SCHEMBL7709557

SCHEMBL7709557

N#Cc1cc2c3c(cccc3c1Cl)C(=O)N(OCc1ccccc1)C2=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP1B1 Q16678 2/20 0.39
HTT P42858 2/20 0.39
RGS12 O14924 1/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
RECQL P46063 1/20 0.39
ATM Q13315 1/20 0.39
CNR1 P21554 3/20 0.36
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 2/20 0.35
BCAT2 O15382 1/20 0.35
HPGD P15428 1/20 0.35
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703771 0.83 KMT2A (0.51) MEN1KMT2AMAPTSMN1; SMN2POLB
SCHEMBL7706689 0.82 MEN1 (0.39) MEN1KMT2AMAPTSMN1; SMN2POLB
SCHEMBL7709619 0.81 MEN1 (0.39) MEN1KMT2AMAPTSMN1; SMN2POLB
SCHEMBL7703898 0.74 CTSL (0.39)
SCHEMBL7712257 0.74 MEN1 (0.46) MEN1KMT2AMAPTPOLBGAA
SCHEMBL7712197 0.73 CYP1B1 (0.65) MEN1KMT2AMAPTPOLBCYP1B1
SCHEMBL7703721 0.72 CYP1B1 (0.46) MEN1KMT2AMAPTPOLBCYP1B1
SCHEMBL7709360 0.72 KMT2A (0.43) MEN1KMT2AMAPTPOLBGAA
SCHEMBL7703787 0.72 KMT2A (0.43) MEN1KMT2AMAPTPOLBGAA
SCHEMBL7706791 0.72 PRMT1 (0.60) MEN1KMT2AMAPTPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed