SCHEMBL7710137

SCHEMBL7710137

CCOC(=O)c1ccc(N(CC)c2ccc3c(c2)C(C)(C)CC(=O)N3C(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARA P10276 5/20 0.50
RARB P10826 5/20 0.50
RARG P13631 2/20 0.50
RXRA P19793 12/20 0.43
RXRB P28702 4/20 0.43
RXRG P48443 4/20 0.43
MAPK1 P28482 1/20 0.41
WRN Q14191 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703983 0.89 RARA (0.51) RARARARBRARGRXRAMAPK1
SCHEMBL8122120 0.88 RARA (0.64) RARARARBRARGRXRARXRB
SCHEMBL7710045 0.82 RARA (0.52) RARARARBRARGRXRAMAPK1
SCHEMBL8634168 0.82 RARB (0.74) RARARARBRARGRXRAMAPK1
SCHEMBL8115004 0.82 RARA (0.69) RARARARBRARGRXRARXRB
SCHEMBL7703980 0.79 MEN1 (0.50) RARARARBRARGRXRAMAPK1
SCHEMBL7710145 0.79 RARA (0.48) RARARARBRARGRXRAMAPK1
SCHEMBL7710141 0.78 RARA (0.47) RARARARBRARGRXRAMAPK1
SCHEMBL8634937 0.77 RARB (0.74) RARARARBRARGRXRAMAPK1
SCHEMBL7712306 0.76 RARA (0.61) RARARARBRARGRXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228042-A2 TETRAHYDROQUINOLINE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2002-08-07 EP disclosed
WO-2001012606-A2 TETRAHYDROQUINOLINE DERIVATIVES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 2001-02-22 WO disclosed
US-6127382-A AN ANTIPROLIFERATIVE AGENT FOR TREATING SKIN-RELATED DISEASES, AN ANTITUMOR AGENT TREATING CANCER, AN ANTIINFLAMMATORY AGENT TREATING PULMONARY FIBROSIS, ILEITIS, COLITIS AND KROHN'S DISEASE ALLERGAN SALES, INC. (US) 2000-10-03 US disclosed