SCHEMBL7712835

SCHEMBL7712835

CCc1ccc(-c2ccc3c(c2)CNC3=O)c(OCCC(C)C)c1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.40
MAPKAPK2 P49137 1/20 0.40
DAPK3 O43293 1/20 0.40
NTRK1 P04629 1/20 0.40
PIM1 P11309 1/20 0.40
FLT3 P36888 1/20 0.40
ROCK1 Q13464 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
PRKCI P41743 1/20 0.39
MGAM O43451 2/20 0.38
GAA P10253 2/20 0.38
SI P14410 2/20 0.38
MGAM2 Q2M2H8 2/20 0.38
BRAF P15056 1/20 0.37
POLQ O75417 1/20 0.36
HSD17B1 P14061 1/20 0.35
TBK1 Q9UHD2 1/20 0.35
PIK3CD O00329 1/20 0.35
AKT1 P31749 1/20 0.35
TGFBR1 P36897 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2591201 0.88 MGAM (0.43) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL2585698 0.78 GSK3B (0.42) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL14737126 0.77 POLQ (0.39) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL7712508 0.77 MAPKAPK2 (0.38) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL2593088 0.76 GSK3B (0.41) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL14737558 0.75 POLQ (0.37) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL14736569 0.75 POLQ (0.37) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL26029646 0.75 TDP1 (0.43) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL7713989 0.74 POLQ (0.37) GSK3BMAPKAPK2DAPK3NTRK1PIM1
SCHEMBL2589137 0.74 GSK3B (0.40) GSK3BMAPKAPK2DAPK3NTRK1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011134468-A1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2011-11-03 WO disclosed