SCHEMBL7712508

SCHEMBL7712508

CCc1ccc(-c2ccc3c(c2)CNC3=O)c(OCc2ccc(S(N)(=O)=O)cc2)c1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.38
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA9 Q16790 4/20 0.36
CA12 O43570 1/20 0.36
DAPK3 O43293 1/20 0.36
NTRK1 P04629 1/20 0.36
PIM1 P11309 1/20 0.36
FLT3 P36888 1/20 0.36
GSK3B P49841 1/20 0.36
ROCK1 Q13464 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
PTGS2 P35354 5/20 0.36
PTGS1 P23219 2/20 0.36
AKT1 P31749 1/20 0.35
PRKCI P41743 1/20 0.35
TARS1 P26639 1/20 0.35
CA7 P43166 3/20 0.35
CA4 P22748 1/20 0.35
CA14 Q9ULX7 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592812 0.90 CA1 (0.41) MAPKAPK2CA1CA2CA9CA12
SCHEMBL2594294 0.85 AKT1 (0.36) MAPKAPK2CA1CA2CA9CA12
SCHEMBL2588115 0.81 PTGS2 (0.39) MAPKAPK2DAPK3NTRK1PIM1FLT3
SCHEMBL2593103 0.80 TARS1 (0.40) MAPKAPK2CA1CA2CA9CA12
SCHEMBL2584393 0.77 PDE4A (0.37) MAPKAPK2DAPK3NTRK1PIM1FLT3
SCHEMBL7712835 0.77 GSK3B (0.40) MAPKAPK2DAPK3NTRK1PIM1FLT3
SCHEMBL2588546 0.75 PRF1 (0.51) MAPKAPK2DAPK3NTRK1PIM1FLT3
SCHEMBL7711917 0.75 MAOA (0.45) PTGS2PTGS1
SCHEMBL2584262 0.73 SLC6A4 (0.42) MAPKAPK2DAPK3NTRK1PIM1FLT3
SCHEMBL14737565 0.73 MAOA (0.45) CA1CA2CA9CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011134468-A1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2011-11-03 WO disclosed