SCHEMBL7714532

SCHEMBL7714532

COC(=O)Cc1ccc(NCC(C)N(CC(O[Si](C)(C)C(C)(C)C)c2cccc(Cl)c2)C(=O)OC(C)(C)C)cc1F

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.32
ADRB3 P13945 5/20 0.32
ADRB1 P08588 4/20 0.32
P2RX3 P56373 1/20 0.31
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 2/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714670 0.94 ADRB2 (0.33) ADRB2ADRB3ADRB1MAPTNPSR1
SCHEMBL7716950 0.92 ADRB2 (0.32) ADRB2ADRB3ADRB1
SCHEMBL7709011 0.92 NR1H2 (0.32) ADRB2ADRB3ADRB1
SCHEMBL7712721 0.89 RPS6KB1 (0.30)
SCHEMBL7708894 0.86 ADRB2 (0.32) ADRB2ADRB3ADRB1
SCHEMBL7714945 0.85 CYP3A4 (0.30) CYP3A4
SCHEMBL7714622 0.84
SCHEMBL7714803 0.84 PDCD1 (0.33) MAPT
SCHEMBL8586129 0.83 ADRB3 (0.37) ADRB2ADRB3ADRB1MAPT
SCHEMBL8586133 0.83 ADRB3 (0.37) ADRB2ADRB3ADRB1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865421-B1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS AGONISTS OF ATYPICAL BETA-ADRENOCEPTORS GLAXO GROUP LTD (GB) 2002-03-27 EP disclosed
US-6048872-A DIETETICS; ANTIDIABETIC AGENTS; CARDIOVASCULAR DISORDERS; GASTROINTESTINAL DISORDERS GLAXO WELLCOME INC. (US) 2000-04-11 US disclosed