SCHEMBL7714927

SCHEMBL7714927

CC(C)[Si](Oc1ccc2cccc(NC(=O)OC(C)(C)C)c2c1)(C(C)C)C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.43
PLAU P00749 1/20 0.43
NQO2 P16083 1/20 0.39
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
KDM4E B2RXH2 2/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRB2 P47870 1/20 0.38
KMT2A Q03164 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
BRD9 Q9H8M2 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709234 0.85 TRPV1 (0.44) TRPV1PLAUNQO2HPGDALDH1A1
SCHEMBL14433303 0.83 TRPV1 (0.53) TRPV1PLAUHPGDALDH1A1KDM4E
SCHEMBL6469664 0.81 TRPV1 (0.46) TRPV1PLAUNQO2HPGDALDH1A1
SCHEMBL1963401 0.80 MTNR1A (0.50) TRPV1PLAUNQO2HPGDALDH1A1
SCHEMBL7717631 0.80 GAA (0.36) NQO2HPGDALDH1A1KDM4EGLA
SCHEMBL2412766 0.80 POLB (0.42) ALDH1A1GAAMAPTKMT2ABRD9
SCHEMBL487112 0.79 TRPV1 (0.44) TRPV1PLAUNQO2HPGDALDH1A1
SCHEMBL6432988 0.79 NQO2 (0.47) NQO2HPGDALDH1A1KDM4EGLA
SCHEMBL2771446 0.79 CYP17A1 (0.48) RXFP1GAANPC1RAB9A
SCHEMBL14134840 0.78 MTNR1A (0.51) TRPV1PLAUHPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed