SCHEMBL7717142

SCHEMBL7717142

[O]CCCc1cccnn1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CTDSP1 Q9GZU7 1/20 0.40
P2RX7 Q99572 1/20 0.36
VNN1 O95497 1/20 0.36
CES1 P23141 1/20 0.35
GOT1 P17174 1/20 0.33
HRH1 P35367 2/20 0.33
CYP2C9 P11712 1/20 0.33
NAMPT P43490 1/20 0.33
CHRM1 P11229 1/20 0.33
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KCNH2 Q12809 1/20 0.31
NAAA Q02083 1/20 0.31
BRD4 O60885 1/20 0.31
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6241871 0.87
SCHEMBL18854185 0.87 CYP1A2 (0.44) CYP1A2CTDSP1P2RX7VNN1CES1
SCHEMBL3079246 0.82 CYP1A2 (0.47) CYP1A2CTDSP1P2RX7VNN1CES1
SCHEMBL7718075 0.79 CYP1A2 (0.40) CYP1A2CTDSP1P2RX7VNN1CES1
SCHEMBL4722142 0.79 CYP1A2 (0.40) CYP1A2CTDSP1P2RX7VNN1CES1
SCHEMBL29221868 0.79 HRH1 (0.48) CYP1A2CTDSP1P2RX7VNN1GOT1
SCHEMBL20099842 0.79 CYP1A2 (0.43) CYP1A2CTDSP1P2RX7VNN1CES1
SCHEMBL4171814 0.79 KCNH2 (0.48) CYP1A2CTDSP1HRH1CHRM1KCNH2
SCHEMBL344825 0.78
SCHEMBL655646 0.78 KCNH2 (0.57) CYP1A2CTDSP1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002087587-A2 4-AMINOSULFONYLQUINAZOLINES AND -QUINOLINES AS TYROSINE KINASE INHIBITORS CELLTECH R & D LIMITED (GB) 2002-11-07 WO disclosed