SCHEMBL7717411

SCHEMBL7717411

CCCNc1cc2[nH]c(=O)c(C)c(C(F)(F)F)c2cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.51
MMP2 P08253 2/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
TRPA1 O75762 1/20 0.33
CYP1A2 P05177 1/20 0.33
PARP1 P09874 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
ALDH1A1 P00352 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 2/20 0.31
MAPT P10636 2/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
TSHR P16473 2/20 0.31
HSD17B10 Q99714 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1771600 0.78 AR (0.77) AR
SCHEMBL7709128 0.75 AR (0.34) ARALDH1A1KDM4EMAPTGLA
SCHEMBL1772197 0.70 AR (0.62) AR
SCHEMBL1771533 0.68 AR (1.00) AR
SCHEMBL1771203 0.66 AR (0.45) AR
SCHEMBL2833045 0.64 DAO (0.53) CYP1A2PARP1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL18893379 0.63 IDO1 (0.36) ARTRPA1CYP1A2ALDH1A1SMN1; SMN2
SCHEMBL1771709 0.62 AR (0.61) AR
SCHEMBL1771723 0.62 AR (0.78) AR
SCHEMBL1771664 0.59 AR (1.00) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212303-A2 BICYCLIC ANDROGEN AND PROGESTERONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2002-06-12 EP disclosed
WO-2001016108-A2 BICYCLIC ANDROGEN AND PROGESTERONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2001-03-08 WO disclosed