SCHEMBL7709128

SCHEMBL7709128

CCCN(C)c1cc2[nH]c(=O)c(C)c(C(F)(F)F)c2cc1F

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.34
DAO P14920 1/20 0.33
MPO P05164 2/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7717411 0.75 AR (0.51) ARKDM4EALDH1A1GLAGAA
SCHEMBL2833045 0.63 DAO (0.53) DAOKDM4EALDH1A1GLAGAA
SCHEMBL20207784 0.59 AKR1B1 (0.44) DAOKDM4EALDH1A1HTT
SCHEMBL5716104 0.57 NR3C2 (0.39) ALDH1A1HTT
SCHEMBL31193836 0.57 AOC1 (0.39) AR
SCHEMBL1772197 0.57 AR (0.62) AR
SCHEMBL21324919 0.56 CYP1A2 (0.38) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL6680406 0.56 KDM4E (0.50) MPOKDM4EALDH1A1GAAMAPT
SCHEMBL4287768 0.56 CA12 (0.41) ARDAOKDM4EALDH1A1MAPT
SCHEMBL17774951 0.56 HCAR3 (0.35) MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212303-A2 BICYCLIC ANDROGEN AND PROGESTERONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2002-06-12 EP disclosed
WO-2001016108-A2 BICYCLIC ANDROGEN AND PROGESTERONE RECEPTOR MODULATOR COMPOUNDS AND METHODS LIGAND PHARMACEUTICALS INCORPORATED (US) 2001-03-08 WO disclosed