SCHEMBL7720550

SCHEMBL7720550

O=C(NCC(F)(F)F)OC1(CCCCN2CCN(c3ccc(-c4ccccc4)cc3)CC2)c2ccccc2-c2ccc(Cl)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.43
DRD4 P21917 6/20 0.43
DRD3 P35462 5/20 0.40
ADRA1A P35348 2/20 0.40
MTTP P55157 2/20 0.40
CHRM2 P08172 1/20 0.40
ADRA2A P08913 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
PTGS1 P23219 1/20 0.40
SLC6A2 P23975 1/20 0.40
OPRM1 P35372 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KCNH2 Q12809 1/20 0.40
MTR Q99707 1/20 0.40
HTR7 P34969 4/20 0.40
HTR1A P08908 1/20 0.40
FAAH O00519 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7720317 0.94 DRD2 (0.47) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7716462 0.93 DRD3 (0.43) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7721461 0.92 HTR2A (0.41) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7720585 0.91 DRD3 (0.41) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7720551 0.90 DRD3 (0.43) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7720477 0.88 DRD3 (0.44) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7723358 0.88 DRD2 (0.46) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7723388 0.88 DRD3 (0.42) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7723394 0.87 DRD3 (0.44) DRD2DRD4DRD3ADRA1AMTTP
SCHEMBL7721420 0.87 DRD3 (0.47) DRD2DRD4DRD3ADRA1AMTTP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228053-A1 SUBSTITUTED PIPERAZINE DERIVATIVES, THE PRODUCTION AND USE THEREOF AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) Boehringer Ingelheim Pharma KG (DE) 2002-08-07 EP disclosed
WO-2001021604-A1 SUBSTITUTED PIPERAZINE DERIVATIVES, THE PRODUCTION THEREOF AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE-TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-03-29 WO disclosed