SCHEMBL7721956

SCHEMBL7721956

COC(=O)[C@@H]1CC(CN(C=O)OC(C)(C)C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 1/20 0.34
PTPN1 P18031 1/20 0.34
MMP2 P08253 2/20 0.33
ANPEP P15144 2/20 0.33
TGM2 P21980 2/20 0.33
P2RX3 P56373 2/20 0.33
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CCNT1 O60563 1/20 0.30
CDK9 P50750 1/20 0.30
F13A1 P00488 1/20 0.30
TGM1 P22735 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7729539 0.92 NR1H2 (0.38) NR1H2TGM2CYP1A2POLBCYP3A4
SCHEMBL7722084 0.88 NR1H2 (0.39) NR1H2TGM2CYP1A2POLBCYP3A4
SCHEMBL7721995 0.88 NR1H2 (0.39) NR1H2TGM2CYP1A2POLBCYP3A4
SCHEMBL7729001 0.81 NR1H2 (0.44) NR1H2
SCHEMBL31000687 0.79 NR1H2 (0.40) NR1H2NR1H3PTPN1MMP2ANPEP
SCHEMBL9601879 0.79 NR1H2 (0.40) NR1H2NR1H3PTPN1MMP2ANPEP
SCHEMBL29851070 0.79 NR1H2 (0.40) NR1H2NR1H3PTPN1MMP2ANPEP
SCHEMBL17317642 0.79 NR1H2 (0.40) NR1H2NR1H3PTPN1MMP2ANPEP
SCHEMBL6185885 0.79 NR1H2 (0.40) NR1H2NR1H3PTPN1MMP2ANPEP
SCHEMBL6184330 0.79 NR1H2 (0.40) NR1H2NR1H3PTPN1MMP2ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed
WO-2000001714-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed