SCHEMBL7722771

SCHEMBL7722771

NCCN1CCN(c2n[nH]c3cc(F)ccc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.43
MAP2K4 P45985 5/20 0.40
HTR1A P08908 3/20 0.39
HTR7 P34969 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTT P42858 2/20 0.39
PARP1 P09874 1/20 0.38
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
MAPK1 P28482 2/20 0.38
MAP2K7 O14733 1/20 0.38
PLK1 P53350 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
MAPKAPK3 Q16644 1/20 0.37
MAPK6 Q16659 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9778524 0.85 HTR2A (0.44) HTR2AHTR1AHTR7KDM4EALDH1A1
SCHEMBL8350202 0.84 MAP2K4 (0.42) HTR2AMAP2K4HTR1AHTR7KDM4E
SCHEMBL9778496 0.83 HTR2A (0.52) HTR2AMAP2K4KDM4EALDH1A1HPGD
SCHEMBL1545286 0.83 HTR2A (0.42) HTR2AMAP2K4HTR1AHTR7KDM4E
SCHEMBL1545504 0.83 ADRA1D (0.44) HTR2AMAP2K4HTR1AHTR7KDM4E
SCHEMBL27263489 0.83 DRD4 (0.49) MAP2K4HTR1AHTR7PLK1DRD2
SCHEMBL1545843 0.82 HTR2A (0.41) HTR2AMAP2K4HTR1AHTR7KDM4E
Hydrochloric Acid SCHEMBL7726743 0.81 HTR2A (0.41) HTR2AMAP2K4HTR1AHTR7KDM4E
SCHEMBL1544905 0.81 ADRA1D (0.49) HTR2AMAP2K4HTR1AHTR7DRD2
SCHEMBL1545365 0.81 PARP1 (0.54) HTR2AHTR1AHTR7KDM4EPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420390-B1 ANALGESIC AGENTS AVENTIS PHARMACEUTICALS INC. 2002-07-16 US disclosed
US-RE37729-E1 4-Heteroaryl-1-piperidinealkylamines and derivatives thereof and their therapeutic utility AVENTIS PHARMACEUTICALS INC. 2002-06-04 US disclosed
US-6251907-B1 1-(aryloxyalkyl)-4-(heteroaryl) piperazines and related compounds useful as antipsychotics and analgesics AVENTIS PHARMACEUTICALS INC. 2001-06-26 US disclosed
US-6001834-A PSYCHOLOGICAL DISORDERS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1999-12-14 US disclosed
US-5965546-A ANTIPSYCHOTIC AND ANALGESIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-10-12 US disclosed
US-5919798-A USEFUL AS ANTIPSYCHOTIC AND ANALGESIC AGENTS. HOECHST MARION ROUSSEL, INC. (US) 1999-07-06 US disclosed
US-5889035-A 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed
US-5889004-A PSYCHOLOGICAL DISORDERS, ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed
US-5874435-A PSYCHOLOGICAL DISORDERS; ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-02-23 US disclosed
US-5854263-A 1- (1,4-benzodioxanyl)alkyl!-3-(heteroaryl) pyrrolidines and related compounds and their therapeutic utility HOECHST MARION ROUSSEL, INC. (US) 1998-12-29 US disclosed
US-5843977-A (3-heteroaryl-1-pyrrolidinyl) alkoxy!-3,4-dihydro-1(2H)-naphthalenones and related compounds and their therapeutic utility HOECHST MARION ROSUEEL, INC. 1998-12-01 US disclosed
US-5843949-A 1-(1H-indolyloxyalkyl)-4-(heteroaryl)piperazines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. 1998-12-01 US disclosed
US-5840727-A ANTIPSYCHOTICS, ANALGESICS AVENTIS PHARMACEUTICALS INC. 1998-11-24 US disclosed
US-5811430-A 1 (2-pyrimidinyloxy) alkyl!-4- (heteroaryl) Piperidines and related compounds and their therapeutic utility HOECHST MARION ROUSSEL, INC. 1998-09-22 US disclosed
US-5811435-A 2- (4-heteroaryl-1-piperidinyl)alkyl!-1,3-dioxanes and related compounds and their therapeutic utility HOECHST MARION RUSSEL, INC. 1998-09-22 US disclosed
US-5776963-A ANTIPSYCHOTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-07-07 US disclosed
US-5589495-A ANTIPSYCHOTIC AGENTS, ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1996-12-31 US disclosed