SCHEMBL7723246

SCHEMBL7723246

C=C[C@@H](CCCNC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.59
GAA P10253 1/20 0.59
KMT2A Q03164 1/20 0.59
TDP1 Q9NUW8 1/20 0.50
CTSK P43235 16/20 0.47
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31483558 0.85 CTSK (0.49) TDP1CTSK
SCHEMBL12893562 0.85 CTSK (0.63) CTSK
SCHEMBL3498473 0.82 CTSK (0.60) MEN1GAAKMT2ATDP1CTSK
SCHEMBL3818710 0.82 CTSK (0.60) MEN1GAAKMT2ATDP1CTSK
SCHEMBL6339388 0.82 MEN1 (0.62) MEN1GAAKMT2ATDP1MAOA
SCHEMBL23009079 0.81 CTSK (0.51) CTSK
SCHEMBL15221109 0.81 CTSK (0.49) CTSK
SCHEMBL24906968 0.81 MEN1 (0.54) MEN1GAAKMT2ATDP1CTSK
SCHEMBL6277041 0.80 MEN1 (0.64) MEN1GAAKMT2ATDP1CTSK
SCHEMBL20738187 0.79 CTSK (0.47) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed
WO-1999037667-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 1999-07-29 WO disclosed