SCHEMBL7729320

SCHEMBL7729320

COC(=O)[C@H]1CC(NC(=O)C(O)C(N)C(=O)OC(C)(C)C)CN1C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 11/20 0.37
PEPD P12955 4/20 0.36
HTRA1 Q92743 1/20 0.36
ANPEP P15144 6/20 0.36
XPNPEP1 Q9NQW7 2/20 0.36
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
PTPN1 P18031 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7727563 0.90 HTRA1 (0.39) MMP2HTRA1ANPEPCYP1A2POLB
SCHEMBL7731684 0.79 BTK (0.46) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL13938227 0.79 MMP2 (0.47) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL7727313 0.79 BTK (0.46) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL13938226 0.79 MMP2 (0.47) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL7727315 0.79 BTK (0.46) MMP2ANPEPNR1H2NR1H3PTPN1
SCHEMBL7727763 0.77 MMP2 (0.36) MMP2PEPDANPEPXPNPEP1NR1H2
SCHEMBL7727758 0.77 MMP2 (0.36) MMP2PEPDANPEPXPNPEP1NR1H2
SCHEMBL7729316 0.77 MMP2 (0.36) MMP2PEPDANPEPXPNPEP1NR1H2
SCHEMBL12651618 0.77 MMP2 (0.43) MMP2ANPEPNR1H2NR1H3PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399629-B1 PYRROLIDINES AND PIPERIDINES FOR TREATING MICROBIAL INFECTIONS BY REDUCING EXPORT OF COADMINISTERED ANTIMICROBIAL AGENT OR COMPOUND SYNTHESIZED BY MICROBES FOR THEIR GROWTH; REDUCING IN VIVO AVAILABILITY MICROCIDE PHARMACEUTICALS, INC. 2002-06-04 US disclosed