SCHEMBL7733272

SCHEMBL7733272

CCN(C(=O)NCc1ccc(F)c(F)c1)C1CCN(OC(=O)C(F)(F)F)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 14/20 0.47
CCR5 P51681 4/20 0.44
CYP1A2 P05177 2/20 0.42
HTR2C P28335 2/20 0.42
CYP2C19 P33261 2/20 0.42
KCNH2 Q12809 2/20 0.42
HTR2B P41595 1/20 0.42
P2RX7 Q99572 1/20 0.41
HRH3 Q9Y5N1 2/20 0.41
ABCB11 O95342 1/20 0.41
ADRB2 P07550 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
DRD1 P21728 1/20 0.41
TBXA2R P21731 1/20 0.41
SLC6A2 P23975 1/20 0.41
GPR183 P32249 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRM1 P35372 1/20 0.41
APLNR P35414 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723311 0.85 CCR5 (0.49) HTR2ACCR5KCNH2
Trifluoroacetic Acid SCHEMBL7733264 0.80 HTR2A (0.46) HTR2ACCR5KCNH2P2RX7SLC6A2
SCHEMBL7732604 0.78 CCR5 (0.51) HTR2ACCR5CYP1A2HTR2CCYP2C19
SCHEMBL7731085 0.76 CCR5 (0.42) HTR2ACCR5CYP1A2HTR2CCYP2C19
SCHEMBL7723375 0.71 CCR5 (0.43) HTR2ACCR5HRH3
SCHEMBL7736000 0.70 CCR5 (0.51) CCR5KCNH2DRD3
SCHEMBL7732190 0.69 HTR2A (0.49) HTR2ACCR5CYP2C19KCNH2P2RX7
SCHEMBL22361694 0.69 HTR2A (0.65) HTR2ACYP1A2HTR2CCYP2C19KCNH2
SCHEMBL14446775 0.66 CCR5 (0.60) HTR2ACCR5
SCHEMBL20766692 0.66 HTR2A (0.60) HTR2ACYP1A2HTR2CCYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399619-B1 PREVENTION AND TREATMENT OF AIDS AND VIRAL INFECTION BY HIV MERCK & CO., INC. 2002-06-04 US disclosed