SCHEMBL7734291

SCHEMBL7734291

CCSC(=N)Nc1ccc(-n2cccc2)c(CN)c1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7734154 0.99 NPC1 (0.31) NPC1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL27514201 0.99 NPC1 (0.31) NPC1ALDH1A1MAPT
SCHEMBL7739655 0.82 KMT2A (0.36) NPC1ALDH1A1MAPTMAPK1
Hydrochloric Acid SCHEMBL7740465 0.82 KMT2A (0.36) NPC1ALDH1A1MAPTMAPK1
SCHEMBL27552471 0.81 HDAC3 (0.33)
Hydrochloric Acid SCHEMBL27564406 0.80 HDAC3 (0.32)
SCHEMBL27494821 0.79 HDAC3 (0.34) NPC1ALDH1A1MAPTMAPK1
SCHEMBL27479175 0.78 HDAC3 (0.41) NPC1ALDH1A1MAPTMAPK1
SCHEMBL27559508 0.78 TSHR (0.35) NPC1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL27544842 0.78 HDAC3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN claimed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US claimed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN claimed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP claimed
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed