SCHEMBL7739655

SCHEMBL7739655

CCSC(=N)Nc1ccc(-n2cccn2)c(CN)c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.36
MEN1 O00255 7/20 0.36
ALDH1A1 P00352 6/20 0.36
MAPT P10636 6/20 0.36
LMNA P02545 5/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
G6PD P11413 1/20 0.34
MPO P05164 4/20 0.34
HTT P42858 1/20 0.33
MDM2 Q00987 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
TSHR P16473 1/20 0.32
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7740465 0.99 KMT2A (0.36) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL7734291 0.82 NPC1 (0.32) ALDH1A1MAPTNPC1MAPK1
Hydrochloric Acid SCHEMBL27514201 0.81 NPC1 (0.31) ALDH1A1MAPTNPC1
Hydrochloric Acid SCHEMBL7734154 0.81 NPC1 (0.31) ALDH1A1MAPTNPC1
Hydrochloric Acid SCHEMBL7738899 0.81 RXFP1 (0.38) KMT2AMEN1ALDH1A1MAPTLMNA
Hydrochloric Acid SCHEMBL7742139 0.81 AAK1 (0.40) KMT2AMEN1ALDH1A1MAPTRAB9A
Hydrochloric Acid SCHEMBL27512818 0.81 TDO2 (0.32)
Hydrochloric Acid SCHEMBL7740435 0.81 TDO2 (0.32)
SCHEMBL7740424 0.80 MEN1 (0.36) KMT2AMEN1ALDH1A1MAPTLMNA
Hydrochloric Acid SCHEMBL7738922 0.77 LMNA (0.32) KMT2AMEN1ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN claimed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US claimed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN claimed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP claimed
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed