SCHEMBL7735910

SCHEMBL7735910

CSc1sc(C(=N)N)cc1C(=O)N(C)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
C1S P09871 4/20 0.54
PLAU P00749 2/20 0.50
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HPGD P15428 2/20 0.48
GAA P10253 1/20 0.48
HSD17B2 P37059 5/20 0.47
HSP90AA1 P07900 2/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HSD17B1 P14061 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6925414 0.99 C1S (0.53) C1SPLAUHDAC3HDAC4HDAC1
SCHEMBL7735241 0.88 C1S (0.53) C1SPLAUHDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL6923914 0.87 C1S (0.52) C1SPLAUHDAC3HDAC4HDAC1
SCHEMBL6925814 0.84 HPGD (0.54) HDAC3HDAC4HDAC1HDAC6HPGD
SCHEMBL7736159 0.78 C1S (0.55) C1SPLAUHDAC3HDAC4HDAC1
SCHEMBL7735938 0.76 C1S (0.53) C1SPLAUHDAC3HDAC4HDAC1
SCHEMBL7736645 0.76 C1S (0.55) C1SPLAU
Hydrochloric Acid SCHEMBL6924633 0.75 C1S (0.52) C1SPLAUHDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL6925651 0.75 C1S (0.54) C1SPLAU
SCHEMBL7359059 0.74 C1S (0.53) C1SPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403633-B2 USEFUL ANTIANGIOGENIC, ANTIARTHRITIC, ANTIINFLAMMATORY, ANTIRESTENOTIC, ANTIINVASIVE, ANTIMETASTIC, ANTIOSTEOPOROTIC, ANTIRETINOPATHIC, CONTRACEPTIVE AND TUMORISTATIC TREATMENT AGENTS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-06-11 US claimed
WO-2000047194-A9 METHODS OF TREATING C1s-MEDIATED DISEASES AND CONDITIONS, AND COMPOUNDS AND COMPOSITIONS THEREFOR DIMENSIONAL PHARM INC (US) 2001-05-31 WO disclosed