SCHEMBL7736904

SCHEMBL7736904

Cn1cncc1C(C)(NC(=O)CCl)c1ccc(C#N)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 2/20 0.42
S1PR1 P21453 1/20 0.42
CACNA1H O95180 4/20 0.41
FNTA P49354 12/20 0.40
FNTB P49356 12/20 0.40
PGGT1B P53609 12/20 0.40
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7220321 0.89 FNTA (0.41) S1PR3S1PR1CACNA1HFNTAFNTB
SCHEMBL7222226 0.88 FNTA (0.41) S1PR3S1PR1CACNA1HFNTAFNTB
SCHEMBL7241410 0.82 FNTA (0.42) S1PR3S1PR1CACNA1HFNTAFNTB
SCHEMBL7673750 0.82 FNTA (0.44) S1PR3S1PR1FNTAFNTBPGGT1B
SCHEMBL7236823 0.81 FNTA (0.42) CACNA1HFNTAFNTBPGGT1B
SCHEMBL7220418 0.79 ALDH1A1 (0.40) S1PR3S1PR1FNTAFNTBPGGT1B
SCHEMBL7222558 0.78 S1PR3 (0.37) S1PR3S1PR1FNTAFNTBPGGT1B
SCHEMBL7672909 0.78 CYP17A1 (0.48) FNTAFNTBPGGT1BCYP17A1CYP3A4
SCHEMBL7222091 0.75 FNTA (0.47) FNTAFNTBPGGT1BCYP11B1CYP11B2
SCHEMBL7228124 0.75 CYP11B1 (0.36) S1PR3S1PR1CACNA1HFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413964-B1 14-AMINO-14-(1-METHYL-1H-IMIDAZOL-5-YL)-8-OXA-2-THIA-1,18 -DIAZATETRACYCLO(16.2.2.1(3,7).1(9,13))TETRACOSA-3(24),4,6, 9(23),10,12-HEXAENE-10-CARBONITRILE 2,2-DIOXIDE, FOR EXAMPLE; USE IN RADIOTHERAPY, CHEMOTHERAPY AS SENSITIZER MERCK & CO., INC. 2002-07-02 US disclosed