SCHEMBL7737243

SCHEMBL7737243

CC(C)(C)[Si](C)(C)Oc1cccc2c1CCCN2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
NUDT1 P36639 5/20 0.34
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
BCHE P06276 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33
GRIA4 P48058 1/20 0.33
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
HTR1A P08908 2/20 0.31
DRD2 P14416 1/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
OPRK1 P41145 1/20 0.31
SRC P12931 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30479656 0.77 PARP1 (0.50) PARP1
SCHEMBL10381392 0.77 PARP1 (0.50) PARP1
SCHEMBL430401 0.76 ADRB2 (0.53) HTR1AADRB2ADRB1OPRK1
SCHEMBL4895504 0.74 EGFR (0.34) HTR1ADRD2
SCHEMBL4793712 0.72 PARP1 (0.46) PARP1
SCHEMBL29588862 0.71 ADRB2 (0.52) HTR1AADRB2ADRB1
SCHEMBL2487204 0.71 ADRB2 (0.52) HTR1AADRB2ADRB1
SCHEMBL3376891 0.71 ADRB2 (0.34) S1PR1S1PR3HTR1AADRB2ADRB1
Hydrochloric Acid SCHEMBL5732143 0.71 PARP1 (0.45) PARP1
SCHEMBL4703624 0.71 PRMT5 (0.40) PARP1NUDT1PRMT5WDR77GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407096-B1 1,4-BENZOTHIAZINE AND 1,4-BENZOXAZINE DERIVATIVES; HYPOTENSIVE, ANTIISCHEMIC, ANTIALLERGEN, ANTIASTHMATIC AND ANTICOAGULANT AGENTS; CARDIOVASCULAR DISORDERS TORAY INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1028113-A1 FUSED BENZENE HETEROCYCLE DERIVATIVES AND UTILIZATION THEREOF TORAY INDUSTRIES, INC. (JP) 2000-08-16 EP disclosed