SCHEMBL7738852

SCHEMBL7738852

COC(=O)c1ccc(C#Cc2ccc(-c3ccc(OC)cc3)cc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.70
CA2 P00918 2/20 0.70
MAPT P10636 4/20 0.57
KMT2A Q03164 2/20 0.57
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
PTPN11 Q06124 1/20 0.55
APP P05067 3/20 0.53
NPC1 O15118 2/20 0.51
LMNA P02545 1/20 0.51
ACACB O00763 1/20 0.50
GRM3 Q14832 1/20 0.49
RAB9A P51151 2/20 0.49
CA12 O43570 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738854 1.00 CA1 (0.70) CA1CA2MAPTKMT2AKDM4E
SCHEMBL269558 0.89 CA1 (0.88) CA1CA2MAPTKMT2AKDM4E
SCHEMBL16604876 0.89 CA1 (0.88) CA1CA2MAPTKMT2AKDM4E
SCHEMBL3001548 0.88 CA1 (0.72) CA1CA2MAPTKMT2AKDM4E
SCHEMBL69268 0.86 PTPN11 (0.69) CA1CA2MAPTKMT2AKDM4E
SCHEMBL7738912 0.85 CA1 (0.69) CA1CA2MAPTKDM4EPTPN11
SCHEMBL13139895 0.85 TDP1 (0.69) CA1CA2MAPTKMT2AKDM4E
SCHEMBL13139896 0.85 TDP1 (0.69) CA1CA2MAPTKMT2AKDM4E
SCHEMBL7738900 0.85 CA1 (0.69) CA1CA2MAPTKDM4EPTPN11
SCHEMBL20252721 0.84 CA1 (0.60) CA1CA2MAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743777-B1 TRISPHENYL ACYL DERIVATIVES OF THE ECHINOCANDIN CLASS; CANDIDA ALBICANS; ANTIFUNGAL AND ANTIPARASITIC; CYCLIC HEXAPEPTIDES HAVING UNIQUE SIDE CHAIN ACYL GROUP ELI LILLY AND COMPANY 2004-06-01 US disclosed