SCHEMBL7739635

SCHEMBL7739635

CC(C)(C)OC(=O)N(Cc1cc(NC(N)=S)ccc1-n1cccc1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
GAA P10253 2/20 0.35
NR1I3 Q14994 3/20 0.35
KMT2A Q03164 3/20 0.34
CYP1A2 P05177 1/20 0.33
MAPK1 P28482 1/20 0.33
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
GRM2 Q14416 1/20 0.32
MEN1 O00255 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPY2R P49146 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675178 0.85 KDM4E (0.44) ALDH1A1GAANR1I3KMT2AMAPK1
SCHEMBL6678474 0.84 ALDH1A1 (0.39) ALDH1A1GAAKMT2ACYP1A2MAPT
SCHEMBL6675695 0.84 ALDH1A1 (0.39) ALDH1A1GAAKMT2ACYP1A2MAPT
SCHEMBL6675941 0.84 KDM4E (0.43) ALDH1A1GAANR1I3KMT2ACYP1A2
SCHEMBL6681804 0.83 GRM2 (0.38) ALDH1A1GAAKMT2ACYP1A2MAPT
SCHEMBL6678436 0.83 ALDH1A1 (0.40) ALDH1A1GAAKMT2ANPC1
SCHEMBL6676380 0.82 ALDH1A1 (0.37) ALDH1A1GAAKMT2ACYP1A2MAPT
SCHEMBL6682248 0.82 ALDH1A1 (0.40) ALDH1A1GAAKMT2ACYP1A2MAPT
SCHEMBL6679793 0.82 ALDH1A1 (0.35) ALDH1A1GAANR1I3KMT2ACYP1A2
SCHEMBL7742143 0.82 NR1I3 (0.33) ALDH1A1GAANR1I3KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed