SCHEMBL7740701

SCHEMBL7740701

COC(=O)N1CCc2nc[nH]c(=O)c2C1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
SCN9A Q15858 1/20 0.42
PDGFRB P09619 1/20 0.39
F12 P00748 3/20 0.39
MTHFD2 P13995 4/20 0.37
SRC P12931 3/20 0.34
EGFR P00533 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
RBP4 P02753 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2799009 0.86 MAPT (0.48) KDM4ERXFP1SCN9AF12MAPT
SCHEMBL34464199 0.83 SCN9A (0.42) KDM4ERXFP1SCN9AMTHFD2SRC
SCHEMBL2505488 0.79 PARP1 (0.42) KDM4ERXFP1SCN9AF12MAPT
SCHEMBL20738661 0.77 KDM4E (0.41) KDM4ERXFP1SCN9ASRCMAPT
SCHEMBL2795751 0.75 PARP1 (0.51) KDM4ERXFP1F12MAPTMAPK1
SCHEMBL8485777 0.75 CYP2C19 (0.39) SRCEGFR
SCHEMBL12321214 0.74 MTHFD2 (0.61) MTHFD2HPGDMAPK1
SCHEMBL2792908 0.73 DDB1 (0.43) KDM4EMAPTMAPK1
SCHEMBL31214426 0.72 SRC (0.35) KDM4ERXFP1SCN9AMTHFD2SRC
SCHEMBL13654278 0.72 SRC (0.35) KDM4ERXFP1SCN9ASRCEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414157-B1 COMPOUNDS HAVING HIGH AFFINITY FOR 5-HT1B AND 5-HT1C SEROTONIN RECEPTOR; ANTIDEPRESSANTS ABBOTT LABORATORIES 2002-07-02 US disclosed