SCHEMBL7742589

SCHEMBL7742589

N[C@@H](CCCCNC(=O)Cc1cccnc1)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.62
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
FES P07332 1/20 0.49
RET P07949 1/20 0.49
MARK3 P27448 1/20 0.49
TYK2 P29597 1/20 0.49
FLT4 P35916 1/20 0.49
SYK P43405 1/20 0.49
CLK2 P49760 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
LMNA P02545 1/20 0.48
NAPRT Q6XQN6 1/20 0.48
ERCC1 P07992 1/20 0.47
ERCC4 Q92889 1/20 0.47
PTAFR P25105 5/20 0.46
GAA P10253 2/20 0.46
TRPV1 Q8NER1 1/20 0.46
FOLH1 Q04609 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31268378 1.00 EPHX2 (0.62) EPHX2CYP1A2CYP3A4CYP2C9FES
SCHEMBL2234907 0.96 EPHX2 (0.64) EPHX2CYP1A2CYP3A4CYP2C9FES
SCHEMBL2234915 0.96 EPHX2 (0.64) EPHX2CYP1A2CYP3A4CYP2C9FES
SCHEMBL1768899 0.91 EPHX2 (0.70) EPHX2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL2238031 0.91 EPHX2 (0.70) EPHX2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL31258254 0.88 CYP3A4 (0.55) EPHX2CYP1A2CYP3A4CYP2C9FES
SCHEMBL8235888 0.88 CYP3A4 (0.55) EPHX2CYP1A2CYP3A4CYP2C9FES
SCHEMBL3448812 0.86 TRPV1 (0.61) GAATRPV1HPGDATM
SCHEMBL31268357 0.85 GAA (0.50) EPHX2GAATRPV1FOLH1HPGD
SCHEMBL10701360 0.84 EPHX2 (0.58) EPHX2CYP1A2CYP3A4CYP2C9FES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0822827-A4 ANTAGONISTS OF LHRH UNIV TEXAS (US) 2001-07-11 EP disclosed
EP-0822827-A1 ANTAGONISTS OF LHRH BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1998-02-11 EP disclosed
WO-1996033729-A1 ANTAGONISTS OF LHRH BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1996-10-31 WO disclosed