SCHEMBL7743316

SCHEMBL7743316

O=C(O)c1ccccc1-c1cccc(OCc2ccccc2)c1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.60
NR4A2 P43354 2/20 0.60
CTSV O60911 1/20 0.59
CTSL P07711 1/20 0.59
DHODH Q02127 3/20 0.57
CYP4F2 P78329 1/20 0.56
CYP4A11 Q02928 1/20 0.56
MAOB P27338 1/20 0.54
SRD5A2 P31213 1/20 0.53
MCL1 Q07820 2/20 0.53
PTGER1 P34995 2/20 0.53
NR1H4 Q96RI1 1/20 0.53
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
GRM5 P41594 1/20 0.51
TSHR P16473 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7713124 0.88 MRGPRX4 (0.53) MRGPRX4NR4A2CTSVCTSLDHODH
SCHEMBL17796988 0.84 RXRA (0.61) DHODHSMN1; SMN2
SCHEMBL6799282 0.84 MCL1 (0.63) NR4A2DHODHMAOBSRD5A2MCL1
SCHEMBL7080517 0.82 P2RY14 (0.60) MRGPRX4NR4A2CTSVCTSLMAOB
Hydrochloric Acid SCHEMBL9222333 0.82 MCL1 (0.62) NR4A2DHODHMAOBSRD5A2MCL1
SCHEMBL11593773 0.82 P2RY14 (0.60) MRGPRX4NR4A2CTSVCTSLMAOB
Hydrochloric Acid SCHEMBL9222328 0.81 P2RY14 (0.59) MRGPRX4NR4A2CTSVCTSLMAOB
SCHEMBL5112581 0.80 MAOB (0.57) MRGPRX4NR4A2MAOBMCL1PTGER1
SCHEMBL1746678 0.80 FFAR1 (0.76)
SCHEMBL379281 0.79 MAOB (0.67) MRGPRX4NR4A2CYP4F2CYP4A11MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091736-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2001-10-24 EP disclosed
EP-1091736-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-18 EP disclosed
WO-2000001382-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed