SCHEMBL7744481

SCHEMBL7744481

N=C(N)NCCC[C@@H]1NC(=O)[C@H](CCCCNC(=O)CCOCCOCCN)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CC(=O)O)NC(=O)CNC1=O

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.64
ITGAV P06756 4/20 0.64
ITGB1 P05556 1/20 0.64
ITGA5 P08648 1/20 0.64
ITGB5 P18084 3/20 0.55
MC4R P32245 10/20 0.50
MC5R P33032 10/20 0.50
MC3R P41968 10/20 0.50
MC1R Q01726 10/20 0.50
KEAP1 Q14145 1/20 0.50
NFE2L2 Q16236 1/20 0.50
HSP90AB1 P08238 1/20 0.47
ITGA2B P08514 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279121 1.00 ITGB3 (0.64) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL16177741 0.93 ITGB3 (0.61) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL14885782 0.93 ITGB3 (0.61) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL14075719 0.90 ITGB3 (0.54) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL16995729 0.88 ITGB3 (0.58) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL14585830 0.88 ITGB3 (0.53) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL24285406 0.88 ITGB3 (0.60) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL10138534 0.88 ITGB3 (0.60) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL15397366 0.88 ITGB3 (0.60) ITGB3ITGAVITGB1ITGA5ITGB5
SCHEMBL18968795 0.88 ITGB3 (0.55) ITGB3ITGAVITGB1ITGA5ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6537520-B1 Diagnosis and treatment of cancer; kit containing compound having peptide or peptidomimetic functionality that binds to a alpha v beta 3 receptor linked to a chelator BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-03-25 US disclosed