SCHEMBL7744642

SCHEMBL7744642

CCCCC(=O)Nc1oc(-c2ccccc2-c2ccc([N+](=O)[O-])cc2O)nc1-c1ccsc1.CCCCC(=O)Nc1oc(-c2ccccc2-c2cccc(O)c2)nc1-c1ccsc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.38
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
RAB9A P51151 1/20 0.36
FLT1 P17948 2/20 0.36
PKM P14618 1/20 0.36
KIT P10721 1/20 0.36
HPGD P15428 4/20 0.35
FLT4 P35916 1/20 0.35
ADORA1 P30542 2/20 0.35
ADORA2A P29274 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7746647 0.94 KDR (0.41) KDRALDH1A1MAPTMEN1KMT2A
SCHEMBL7744076 0.90 KDR (0.46) KDRALDH1A1MAPTRAB9AFLT1
SCHEMBL7744083 0.86 KDR (0.47) KDRALDH1A1MAPTMEN1KMT2A
SCHEMBL7739077 0.84 KDR (0.42) KDRALDH1A1MAPTMEN1KMT2A
SCHEMBL7739074 0.82 KDR (0.53) KDRRAB9AFLT1FLT4ADORA2A
SCHEMBL7744794 0.82 PKM (0.43) KDRALDH1A1MAPTMEN1KMT2A
SCHEMBL7744763 0.82 KDM4E (0.46) KDRALDH1A1MAPTMEN1KMT2A
SCHEMBL7744098 0.82 FLT1 (0.40) KDRALDH1A1MAPTMEN1KMT2A
SCHEMBL7744776 0.82 MAPT (0.41) ALDH1A1MAPTMEN1KMT2ARAB9A
SCHEMBL7744055 0.81 MEN1 (0.41) ALDH1A1MAPTMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097147-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2001-11-21 EP claimed
EP-1097147-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-05-09 EP claimed
WO-2000002871-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-01-20 WO claimed