SCHEMBL7748830

SCHEMBL7748830

c1cc(-c2cncn2CCCN2CCOCC2)ccn1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NFATC1 O95644 1/20 0.58
GSK3B P49841 1/20 0.58
DYRK1A Q13627 1/20 0.58
MAPK13 O15264 17/20 0.58
MAPK12 P53778 17/20 0.58
MAPK11 Q15759 17/20 0.58
MAPK14 Q16539 17/20 0.58
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25178802 0.76 NFATC1 (0.45) NFATC1GSK3BDYRK1AMAPK13MAPK12
Sb-210313 SCHEMBL4918397 0.73 MAPK13 (1.00) MAPK13MAPK12MAPK11MAPK14
SCHEMBL8860270 0.73 MAPK13 (1.00) MAPK13MAPK12MAPK11MAPK14
SCHEMBL12545505 0.73 CYP11B1 (0.49) MAPK13MAPK12MAPK11MAPK14
SCHEMBL4915601 0.71 MAPK13 (1.00) MAPK13MAPK12MAPK11MAPK14
SCHEMBL20485805 0.71 FYN (0.54) MAPK13MAPK12MAPK11MAPK14
SCHEMBL7091476 0.69 MAPK13 (0.80) MAPK13MAPK12MAPK11MAPK14
SCHEMBL8860588 0.69 MAPK13 (1.00) MAPK13MAPK12MAPK11MAPK14
SCHEMBL4906821 0.69 MAPK13 (1.00) MAPK13MAPK12MAPK11MAPK14
SCHEMBL7076732 0.69 CYP11B1 (0.43) GSK3BMAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906099-A4 A METHOD OF TREATING CANCER MERCK & CO INC (US) 2001-02-07 EP claimed
EP-0906099-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 1999-04-07 EP claimed
WO-1997036587-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1997-10-09 WO claimed