SCHEMBL7752176

SCHEMBL7752176

CCCCOc1cccc2c1C=NC2=N

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP19A1 P11511 1/20 0.43
MCHR1 Q99705 3/20 0.41
PDE5A O76074 2/20 0.39
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
GCGR P47871 2/20 0.36
TLR8 Q9NR97 1/20 0.35
ELANE P08246 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
HTR1B P28222 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7758189 0.72 CYP1A2 (0.34) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
SCHEMBL5155584 0.71 MCHR1 (0.49) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
SCHEMBL19056885 0.70 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
SCHEMBL7921351 0.69 CYP1A2 (0.57) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
SCHEMBL4915520 0.69 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
SCHEMBL28211346 0.69 CYP1A2 (0.49) CYP1A2CYP2C9CYP2C19CYP19A1PDE5A
SCHEMBL9621758 0.68 CYP1A2 (0.61) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
1,2-Dibutoxybenzene SCHEMBL1226749 0.68 CYP1A2 (0.72) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
1,2-Dibutoxybenzene SCHEMBL29428927 0.68 CYP1A2 (0.72) CYP1A2CYP2C9CYP2C19CYP19A1MCHR1
SCHEMBL7756217 0.68 CYP2D6 (0.42) CYP1A2CYP2C9CYP2C19CYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073407-A1 HAIR DYEING METHOD USING AN ALIPHATIC CATIONIC AMINE AND A ALDEHYDE OR KETONE ORQUINONE OR DI-IMINO-ISOINDOLINE OR 3-AMINO-ISO-INDOLONE DERIVATIVES L'OREAL (FR) 2001-02-07 EP disclosed
EP-1056434-A1 DYEING METHOD USING A SPECIFIC CATIONIC DERIVATIVE AND A COMPOUND SELECTED AMONG A SPECIFIC ALDEHYDE, A SPECIFIC KETONE, A QUINONE AND A DI-IMINO-ISOINDOLINE OR 3-AMINO-ISOINDOLONE DERIVATIVE L'OREAL (FR) 2000-12-06 EP disclosed
WO-2000038640-A1 HAIR DYEING METHOD USING AN ALIPHATIC CATIONIC AMINE AND A ALDEHYDE OR KETONE OR QUINONE OR DI-IMINO-ISOINDOLINE OR 3-AMINO-ISO-INDOLONE DERIVATIVES L'OREAL (FR) 2000-07-06 WO disclosed
WO-2000038639-A1 DYEING METHOD USING A SPECIFIC CATIONIC DERIVATIVE AND A COMPOUND SELECTED AMONG A SPECIFIC ALDEHYDE, A SPECIFIC KETONE, A QUINONE AND A DI-IMINO-ISOINDOLINE OR 3-AMINO-ISOINDOLONE DERIVATIVE L'OREAL (FR) 2000-07-06 WO disclosed