SCHEMBL7753365

SCHEMBL7753365

CCOC(=O)CCCOc1ccc2c(c1)CCNC2=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.61
PDE3B Q13370 2/20 0.51
PDE3A Q14432 2/20 0.51
PARP10 Q53GL7 4/20 0.48
PARP11 Q9NR21 4/20 0.48
PDK2 Q15119 2/20 0.47
P2RY12 Q9H244 1/20 0.47
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45
GABRA5 P31644 1/20 0.45
KCNA5 P22460 1/20 0.44
FFAR1 O14842 1/20 0.42
ALDH2 P05091 2/20 0.42
AOC3 Q16853 2/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19574541 0.84 PARP11 (0.55) PARP10PARP11GABRG2GABRB3GABRA5
SCHEMBL22815609 0.83 BRD4 (0.82) BRD4PDE3BPDE3APDK2P2RY12
SCHEMBL21052076 0.81 BRD4 (0.71) BRD4PDE3BPDE3APDK2MAOA
SCHEMBL8682850 0.79 BRD4 (0.61) BRD4PDE3BPDE3APDK2P2RY12
SCHEMBL1036450 0.79 KCNA5 (0.53) PARP10PARP11GABRG2GABRB3GABRA5
SCHEMBL1239440 0.78 PARP11 (0.50) PARP10PARP11GABRG2GABRB3GABRA5
SCHEMBL12502481 0.78 PARP11 (0.48) PARP10PARP11GABRG2GABRB3GABRA5
SCHEMBL9133347 0.77 BRD4 (0.65) BRD4PDE3BPDE3APDK2P2RY12
SCHEMBL11603017 0.76 PDE3B (0.63) BRD4PDE3BPDE3APDK2P2RY12
Hydrochloric Acid SCHEMBL12502617 0.75 PARP11 (0.50) PARP10PARP11GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0725059-B1 2,3-DIAMINOPROPIONIC ACID DERIVATIVE SUMITOMO PHARMA (JP) 2001-01-17 EP disclosed
US-6048854-A ANTICOAGULANTS; ANTICANCER AGENT; WOUND HEALING AGENTS;BONE DISORDERS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-04-11 US disclosed
EP-0725059-A1 2,3-DIAMINOPROPIONIC ACID DERIVATIVE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1996-08-07 EP disclosed