SCHEMBL7753776

SCHEMBL7753776

CC(C)CCN=C(NC#N)Nc1cc(Cl)cc(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 1/20 0.42
TBXAS1 P24557 1/20 0.42
QPCT Q16769 6/20 0.42
NAMPT P43490 7/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KCNJ11 Q14654 3/20 0.38
ABCC9 O60706 2/20 0.38
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7753772 1.00 TBXA2R (0.42) TBXA2RTBXAS1QPCTNAMPTCYP3A4
SCHEMBL8143992 0.85 NAMPT (0.43) QPCTNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL8143994 0.85 NAMPT (0.43) QPCTNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL4260989 0.81 QPCT (0.44) TBXA2RTBXAS1QPCTNAMPTCYP3A4
SCHEMBL4260986 0.81 QPCT (0.44) TBXA2RTBXAS1QPCTNAMPTCYP3A4
SCHEMBL7758049 0.81 QPCT (0.44) TBXA2RTBXAS1QPCTNAMPTCYP3A4
SCHEMBL7758572 0.79 KCNJ11 (0.60) TBXA2RTBXAS1CYP3A4CYP2C9CYP2C19
SCHEMBL7758576 0.79 KCNJ11 (0.60) TBXA2RTBXAS1CYP3A4CYP2C9CYP2C19
SCHEMBL8135713 0.77 NAMPT (0.40) QPCTNAMPTCYP3A4CYP2D6CYP2C9
SCHEMBL8135718 0.77 NAMPT (0.40) QPCTNAMPTCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077933-A1 SUBSTITUTED GUANIDINES AND DIAMINONITROETHENES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2001-02-28 EP disclosed
US-6147098-A USEFUL IN THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM, CARDIOVASCULAR SYSTEM, PULMONARY SYSTEM, GASTROINTESTINAL SYSTEM AND ENDOCRINOLOGIC SYSTEM NOVO NORDISK A/S (DK) 2000-11-14 US disclosed
WO-1999058497-A1 SUBSTITUTED GUANIDINES AND DIAMINONITROETHENES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1999-11-18 WO disclosed