SCHEMBL7757579

SCHEMBL7757579

O=C=Nc1cccc(Cc2ccccc2N=C=O)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.41
TSHR P16473 1/20 0.41
TRPA1 O75762 1/20 0.40
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP1A2 P05177 1/20 0.35
PTPN1 P18031 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
BCL2 P10415 1/20 0.30
BCL2L1 Q07817 1/20 0.30
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2906319 0.94 CYP3A4 (0.40) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL28586403 0.90 CYP3A4 (0.46) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL11211323 0.87 CYP3A4 (0.43) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL510928 0.83 CYP3A4 (0.44) CYP3A4TSHRGABRA1GABRB2CYP1A2
SCHEMBL28037071 0.83 CYP3A4 (0.47) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL387552 0.83 CYP3A4 (0.57) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL29854874 0.83 CYP3A4 (0.57) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL1396327 0.82 CYP3A4 (0.56) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL17912718 0.82 CYP3A4 (0.63) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL27122 0.82 CYP3A4 (0.63) CYP3A4TSHRTRPA1GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024665-B1 DIISOCYANATES OR MIXTURES OF DIISOCYANATES OF THE DIPHENYL-METHANE SERIES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS A SYNTHESIS COMPONENT TO PRODUCE POLYURETHANE PLASTICS ACCORDING TO THE ISOCYANATE-POLYADDITION PROCESS BAYER AG (DE) 1982-05-05 EP claimed
EP-0024665-A1 Diisocyanates or mixtures of diisocyanates of the diphenyl-methane series, process for their preparation and their use as a synthesis component to produce polyurethane plastics according to the isocyanate-polyaddition process BAYER AG (DE) 1981-03-11 EP claimed
EP-1082296-A1 STABILISATION OF ORGANIC POLYISOCYANATES Bayer Aktiengesellschaft (DE) 2001-03-14 EP disclosed
WO-1999048863-A1 STABILISATION OF ORGANIC POLYISOCYANATES BAYER AKTIENGESELLSCHAFT (DE) 1999-09-30 WO disclosed
EP-0445608-B1 Stabilisation of organic polyisocyanates BAYER AG (DE) 1994-06-08 EP disclosed
US-5175349-A Stabilization with hydroxyphenylpropionic acid BAYER AKTIENGESELLSCHAFT (DE) 1992-12-29 US disclosed
EP-0445608-A2 Stabilisation of organic polyisocyanates BAYER AG (DE) 1991-09-11 EP disclosed
US-4761498-A Diisocyanates and diisocyanate mixtures based on diphenylmethane, processes for their production and their use as isocyanate component in the production of polyurethane plastics by the isocyanate polyaddition process BAYER AKTIENGESELLSCHAFT (DE) 1988-08-02 US disclosed
EP-0046556-A1 Diisocyanates or mixtures of diisocyanates of the diphenylmethane class, processes for their preparation, as well as their use as synthesis components in the manufacture of polyurethanes by the isocyanate-polyaddition process BAYER AG (DE) 1982-03-03 EP disclosed
EP-0024665-A1 Diisocyanates or mixtures of diisocyanates of the diphenyl-methane series, process for their preparation and their use as a synthesis component to produce polyurethane plastics according to the isocyanate-polyaddition process BAYER AG (DE) 1981-03-11 EP disclosed