SCHEMBL7759717

SCHEMBL7759717

COc1cc(/N=C(/NC#N)Oc2ccccc2)cc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
KIF11 P52732 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
MAPT P10636 3/20 0.35
CRHR1 P34998 1/20 0.34
IMPDH2 P12268 1/20 0.34
GAA P10253 3/20 0.34
MAPK1 P28482 2/20 0.34
EPHX2 P34913 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ADCY8 P40145 1/20 0.33
ADCY1 Q08828 1/20 0.33
P2RX7 Q99572 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
KDR P35968 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
AKR1C3 P42330 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7759723 1.00 KMT2A (0.53) KMT2AKIF11RXRARXRBRXRG
SCHEMBL7756420 0.91 KMT2A (0.60) KMT2AKIF11MAPTIMPDH2GAA
SCHEMBL7753765 0.87 KMT2A (0.41) KMT2AMAPTIMPDH2GAAADCY8
SCHEMBL7753761 0.87 KMT2A (0.41) KMT2AMAPTIMPDH2GAAADCY8
SCHEMBL7753800 0.83 KMT2A (0.57) KMT2AKIF11MAPTCRHR1GAA
SCHEMBL4037230 0.79 KMT2A (0.72) KMT2AMAPTIMPDH2GAAMAPK1
SCHEMBL7759728 0.77 TMPRSS4 (0.43) MAPTGAAMAPK1EPHX2TMPRSS4
SCHEMBL2088566 0.77 KMT2A (0.59) KMT2AMAPTIMPDH2MAPK1KDM4E
SCHEMBL2088564 0.77 KMT2A (0.59) KMT2AMAPTIMPDH2MAPK1KDM4E
SCHEMBL2087129 0.76 KMT2A (0.80) KMT2AMAPTIMPDH2GAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077933-A1 SUBSTITUTED GUANIDINES AND DIAMINONITROETHENES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2001-02-28 EP disclosed
US-6147098-A USEFUL IN THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM, CARDIOVASCULAR SYSTEM, PULMONARY SYSTEM, GASTROINTESTINAL SYSTEM AND ENDOCRINOLOGIC SYSTEM NOVO NORDISK A/S (DK) 2000-11-14 US disclosed
WO-1999058497-A1 SUBSTITUTED GUANIDINES AND DIAMINONITROETHENES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1999-11-18 WO disclosed