SCHEMBL7760129

SCHEMBL7760129

CCCn1c(=O)c2c(nc(C(C)(C)C)n2Cc2ccccc2)n(CCC(=O)N2CCOCC2)c1=O

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 15/20 0.48
ADORA1 P30542 3/20 0.48
ADORA2A P29274 2/20 0.48
ADORA2B P29275 1/20 0.46
MAOB P27338 2/20 0.46
DPP4 P27487 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958774 0.91 ADORA3 (0.49) ADORA3ADORA1ADORA2AADORA2BMAOB
SCHEMBL7759050 0.85 ADORA3 (0.56) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL7760161 0.85 ADORA3 (0.50) ADORA3ADORA1ADORA2AADORA2BDPP4
SCHEMBL8578130 0.84 ADORA3 (0.53) ADORA3ADORA1ADORA2AADORA2BMAOB
SCHEMBL7759017 0.84 ADORA3 (0.54) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL7969368 0.82 ADORA3 (0.52) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL7970324 0.82 ADORA3 (0.52) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL7759031 0.81 ADORA3 (0.57) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL7759748 0.79 ADORA3 (0.57) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL7759758 0.78 ADORA3 (0.52) ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084123-A1 NOVEL ASYMMETRICALLY SUBSTITUTED XANTHINE DERIVATIVES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS WITH AN ADENOSINE-ANTAGONISTIC EFFECT Boehringer Ingelheim Pharma KG (DE) 2001-03-21 EP disclosed
US-6187780-B1 ANTIDEPRESSANTS, ANTIASTHMATIC AGENTS; MIGRAINE BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-02-13 US disclosed
WO-1999054331-A1 NOVEL ASYMMETRICALLY SUBSTITUTED XANTHINE DERIVATIVES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS WITH AN ADENOSINE-ANTAGONISTIC EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-28 WO disclosed