SCHEMBL7765750

SCHEMBL7765750

O=C1CC(CCN2CCC(c3ccccc3)CC2)(c2ccc(Cl)c(Cl)c2)CN1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.55
TACR1 P25103 18/20 0.52
TACR2 P21452 1/20 0.46
TACR3 P29371 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8840258 0.98 CCR5 (0.54) CCR5TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8483405 0.98 CCR5 (0.54) CCR5TACR1TACR2TACR3
SCHEMBL8991959 0.92 TACR1 (0.63) CCR5TACR1TACR2TACR3
SCHEMBL22901986 0.92 TACR1 (0.63) CCR5TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8840357 0.91 TACR1 (0.62) CCR5TACR1TACR2TACR3
SCHEMBL4631735 0.88 TACR1 (0.47) CCR5TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL7749200 0.86 TACR1 (0.46) CCR5TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL7749206 0.86 TACR1 (0.46) CCR5TACR1TACR2TACR3
SCHEMBL7764193 0.86 TACR1 (0.72) CCR5TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8480218 0.85 TACR1 (0.71) CCR5TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1101757-A1 Heterocyclic compounds as tachykinin receptor antagonists SANOFI-SYNTHELABO (FR) 2001-05-23 EP disclosed
EP-0723959-A1 Heterocyclic compounds as tachykinin receptor antagonists, process for their preparation and pharmaceuticals containing them SANOFI (FR) 1996-07-31 EP disclosed