SCHEMBL7767134

SCHEMBL7767134

CC(=O)OC[C@@H](OC(C)=O)[C@@H](OC(C)=O)[C@@H](COc1ccc(I)cc1)OC(C)=O

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.55
ABCB1 P08183 1/20 0.49
AR P10275 1/20 0.43
POLB P06746 4/20 0.43
MAPK1 P28482 1/20 0.43
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.34
APP P05067 2/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8900805 0.83 TDP1 (0.59) TDP1ABCB1ARPOLBMAPK1
SCHEMBL187068 0.78 TDP1 (0.88) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL15298821 0.78 TDP1 (0.88) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL7154355 0.78 TDP1 (0.88) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL7146329 0.78 TDP1 (0.88) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL7766967 0.75 POLB (0.51) TDP1POLBMAPK1MAPTLMNA
SCHEMBL270042 0.75 TDP1 (0.96) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL2175855 0.75 TDP1 (0.96) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL7149374 0.75 TDP1 (0.96) TDP1ABCB1POLBMAPK1MAPT
SCHEMBL7150717 0.75 TDP1 (0.96) TDP1ABCB1POLBMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741128-B1 Sulphuric acid esters of sugar alcohols for the inhibition of the migration and proliferation of smooth muscle cells of the vascular walls HOFFMANN LA ROCHE (CH) 2001-06-20 EP disclosed
US-5830920-A PREVENTION GROWTH OF SMOOTH MUSCLE CELLS HOFFMANN-LA ROCHE INC. (US) 1998-11-03 US disclosed
EP-0741128-A2 Sulphuric acid esters of sugar alcohols for the inhibition of the migration and proliferation of smooth muscle cells of the vascular walls F. HOFFMANN-LA ROCHE AG (CH) 1996-11-06 EP disclosed