SCHEMBL7767505

SCHEMBL7767505

Cc1ccc2c(c1)C(=O)C(=CO)C2

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 2/20 0.57
MAOA P21397 3/20 0.49
MAOB P27338 3/20 0.49
CES2 O00748 4/20 0.46
TNF P01375 2/20 0.42
ACHE P22303 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7767503 1.00 METAP1 (0.57) METAP1MAOAMAOBCES2TNF
SCHEMBL15698059 0.85 CYP19A1 (0.48) METAP1MAOAMAOBACHE
SCHEMBL7767777 0.79 MAOA (0.49) MAOAMAOBCES2TNFACHE
SCHEMBL1609651 0.79 METAP1 (0.71) METAP1MAOAMAOBACHECA1
SCHEMBL4808970 0.79 MIF (0.61) METAP1MAOAMAOBCES2ACHE
SCHEMBL4808965 0.79 MIF (0.61) METAP1MAOAMAOBCES2ACHE
SCHEMBL12034925 0.78 MAOB (0.69) METAP1MAOAMAOBCES2TNF
SCHEMBL6056920 0.77 METAP1 (0.69) METAP1MAOAMAOBACHECA1
SCHEMBL1512741 0.76 METAP1 (0.67) METAP1MAOAMAOBACHECA1
SCHEMBL6056983 0.76 METAP1 (0.67) METAP1MAOAMAOBACHECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700905-B1 Tricyclic pyrazole derivatives HOFFMANN LA ROCHE (CH) 2001-10-31 EP disclosed
US-5561150-A 1-AMINOALKYL-1,4-DIHYDROINDENO(2,1-C)PYRAZOLES OR 1H-BENZ(G)INDAZOLES; SEROTONIN RECEPTOR ANTAGONISTS; ANTIDEPRESSANTS; NERVOUS SYSTEM, PSYCHOLOGICAL AND GASTROINTESTINAL DISORDERS HOFFMAN-LA ROCHE INC. (US) 1996-10-01 US disclosed
EP-0700905-A1 Tricyclic pyrazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1996-03-13 EP disclosed