SCHEMBL7768948

SCHEMBL7768948

O=C(O)/C=C/c1ccc(OC[C@@H](O)[C@H](O)[C@H](O)[C@@H](O)COc2ccc(/C=C/C(=O)O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.54
ATM Q13315 1/20 0.54
HCAR2 Q8TDS4 2/20 0.47
CA12 O43570 1/20 0.47
AKR1B10 O60218 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
ESR1 P03372 1/20 0.47
CA3 P07451 1/20 0.47
PKM P14618 1/20 0.47
TYR P14679 1/20 0.47
AKR1B1 P15121 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
DPP4 P27487 1/20 0.47
CA5A P35218 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
ESR2 Q92731 1/20 0.47
CA14 Q9ULX7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7769013 0.85 CA12 (0.55) CA12CA1CA2TYRCA7
SCHEMBL3692639 0.83 THRB (0.60) THRBATMHCAR2CA12AKR1B10
SCHEMBL157926 0.83 THRB (0.60) THRBATMHCAR2CA12AKR1B10
SCHEMBL11546773 0.81 CYP1A2 (0.57) THRBATMKDM4EMAPK1ALDH1A1
SCHEMBL11686354 0.80 THRB (0.65) THRBATMHCAR2CA12AKR1B10
SCHEMBL8086432 0.79 THRB (0.55) THRBATMKDM4EMAPK1FFAR1
SCHEMBL8084861 0.79 THRB (0.55) THRBATMHCAR2CA12AKR1B10
SCHEMBL8086431 0.79 THRB (0.55) THRBATMKDM4EMAPK1FFAR1
SCHEMBL31351342 0.79 SRD5A2 (0.58) THRBATMSRD5A2KDM4EMAPK1
SCHEMBL7450494 0.79 HIF1A (0.53) THRBATMKDM4EMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741128-B1 Sulphuric acid esters of sugar alcohols for the inhibition of the migration and proliferation of smooth muscle cells of the vascular walls HOFFMANN LA ROCHE (CH) 2001-06-20 EP disclosed
EP-0741128-A2 Sulphuric acid esters of sugar alcohols for the inhibition of the migration and proliferation of smooth muscle cells of the vascular walls F. HOFFMANN-LA ROCHE AG (CH) 1996-11-06 EP disclosed