SCHEMBL7769665

SCHEMBL7769665

Nc1nc(Sc2ccccc2)c2ncn(CCOCP)c2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.47
CYP2C19 P33261 4/20 0.47
CYP2C9 P11712 3/20 0.47
HIF1A Q16665 3/20 0.47
CYP3A4 P08684 2/20 0.47
ALDH1A1 P00352 1/20 0.47
PHLPP2 Q6ZVD8 1/20 0.47
SLC29A1 Q99808 3/20 0.45
CYP2D6 P10635 2/20 0.41
ADORA2A P29274 3/20 0.39
HK1 P19367 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
MGMT P16455 1/20 0.37
POLB P06746 2/20 0.36
ADORA1 P30542 1/20 0.36
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7770897 0.87 NSD3 (0.45) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7771327 0.86 CYP1A2 (0.42) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7770867 0.86 DHFR (0.45) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7769662 0.86 CYP2C19 (0.44) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7769858 0.86 SLC29A1 (0.46) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7769647 0.85 SLC29A1 (0.41) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7769599 0.85 SLC29A1 (0.40) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7770913 0.84 SLC29A1 (0.43) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7127274 0.84 FGFR1 (0.53) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7769183 0.84 SLC29A1 (0.46) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785208-B1 Phosphonate nucleotide compounds MITSUBISHI CHEM CORP (JP) 2001-03-21 EP claimed
EP-0785208-A1 Phosphonate nucleotide compounds MITSUBISHI CHEMICAL CORPORATION (JP) 1997-07-23 EP claimed
EP-2846788-A1 USE OF COMPOUNDS FOR THE TREATMENT OF PAIN Akron Molecules AG (AT) 2015-03-18 EP disclosed
WO-2013167743-A1 USE OF COMPOUNDS FOR THE TREATMENT OF PAIN AKRON MOLECULES GMBH (AT) 2013-11-14 WO disclosed
EP-0785208-B1 Phosphonate nucleotide compounds MITSUBISHI CHEM CORP (JP) 2001-03-21 EP disclosed
EP-0785208-A1 Phosphonate nucleotide compounds MITSUBISHI CHEMICAL CORPORATION (JP) 1997-07-23 EP disclosed