SCHEMBL7773292

SCHEMBL7773292

Cc1cc(C(=O)O)cc2c1S(=O)(=O)NC2=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.42
CA12 O43570 13/20 0.38
CA9 Q16790 13/20 0.38
CA2 P00918 12/20 0.38
CA7 P43166 7/20 0.38
CA1 P00915 5/20 0.37
CA4 P22748 3/20 0.37
TPMT P51580 1/20 0.37
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
BCHE P06276 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
KMT2A Q03164 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
GRIK1 P39086 1/20 0.35
GRIA1 P42261 1/20 0.35
GRIA2 P42262 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11677692 0.78 CA12 (0.54) CA12CA9CA2CA7CA1
SCHEMBL18726067 0.76 CA12 (0.41) CA12CA9CA2CA7CA1
SCHEMBL7656172 0.70 CHEK1 (0.57) TTRCA12CA9CA2CA7
SCHEMBL8285740 0.69 TTR (0.40) TTRCA12CA9CA2CA7
SCHEMBL3399246 0.68 CA12 (0.59) CA12CA9CA2CA7CA1
SCHEMBL29643009 0.68 CA12 (0.59) CA12CA9CA2CA7CA1
SCHEMBL3259642 0.67 CA1 (0.50) CA12CA9CA2CA7CA1
SCHEMBL1572119 0.64 TPMT (0.59) TTRCA12CA9CA2CA7
SCHEMBL8047467 0.64 TPMT (0.59) TTRCA12CA9CA2CA7
SCHEMBL1081860 0.63 CA12 (0.50) CA12CA9CA2CA7CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775124-B1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AG (DE) 2001-09-19 EP claimed
EP-0775124-A1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1997-05-28 EP claimed
WO-1996005184-A1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1996-02-22 WO claimed
EP-0775124-B1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AG (DE) 2001-09-19 EP disclosed
EP-0775124-B1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AG (DE) 2001-09-19 EP disclosed
CN-1059207-C Herbicidal saccharin carboxylic and its ester defivatives and method for their prep. BASF AG (DE) 2000-12-06 CN disclosed
US-5863864-A REACTING CORRESPONDING BROMO- OR IODO-SUBSTITUTED SACCHARIN DERIVATIVES IN THE PRESENCE OF A PALLADIUM, NICKEL, COBALT OR RHODIUM TRANSITION METAL CATALYST AND OF A BASE WITH CARBON MONOXIDE AND WATER OR A C1-C6 ALCOHOL BASF AKTIENGESELLSCHAFT (DE) 1999-01-26 US disclosed
EP-0775124-A1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1997-05-28 EP disclosed
EP-0775124-A1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1997-05-28 EP disclosed
WO-1996005184-A1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1996-02-22 WO disclosed
WO-1996005184-A1 HERBICIDAL SACCHARIN CARBOXYLIC ACID DERIVATIVES AND METHOD FOR THEIR PREPARATION BASF AKTIENGESELLSCHAFT (DE) 1996-02-22 WO disclosed