SCHEMBL7775249

SCHEMBL7775249

O=C(O)[C@@H]1CC[C@@H](c2cccc(O)c2)N1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.52
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
SCN3A Q9NY46 2/20 0.43
CYP2C19 P33261 3/20 0.41
DPP4 P27487 1/20 0.40
DHFR P00374 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7773300 1.00 KCNH2 (0.52) KCNH2CHRNB4CHRNA3SCN3ACYP2C19
SCHEMBL7769177 1.00 KCNH2 (0.52) KCNH2CHRNB4CHRNA3SCN3ACYP2C19
SCHEMBL7769176 1.00 KCNH2 (0.52) KCNH2CHRNB4CHRNA3SCN3ACYP2C19
SCHEMBL2038087 0.84 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4
SCHEMBL1226045 0.83 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4
SCHEMBL8513273 0.83 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4
SCHEMBL5696388 0.83 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4
SCHEMBL197425 0.83 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4
SCHEMBL135105 0.83 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4
SCHEMBL135106 0.83 KCNH2 (0.56) KCNH2SCN3ACYP2C19DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723974-B1 Derivatives of mercaptoalkanoyldipeptides, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-08-16 EP disclosed
US-5741781-A NEUTRAL ENDOPEPTIDASE AND ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS ADIR ET COMPAGNIE (FR) 1998-04-21 US disclosed
EP-0723974-A1 Derivatives of mercaptoalkanoyldipeptides, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-07-31 EP disclosed