SCHEMBL7775417

SCHEMBL7775417

NC(Cc1nc2ccc(F)cc2s1)N1CCN(c2ncccn2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.45
DRD4 P21917 3/20 0.45
DRD3 P35462 3/20 0.45
HTR1A P08908 2/20 0.45
HTR7 P34969 2/20 0.45
SLC6A2 P23975 2/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2C P18825 1/20 0.45
ADRA1A P35348 1/20 0.45
HRH1 P35367 1/20 0.45
HTR2B P41595 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
DPP4 P27487 1/20 0.44
DPP8 Q6V1X1 1/20 0.44
DPP9 Q86TI2 1/20 0.44
DPP7 Q9UHL4 1/20 0.44
HTR2A P28223 1/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7775355 0.92 KDM4E (0.42) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL7856234 0.91 OGA (0.43) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL7769242 0.89 OGA (0.42) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL7773438 0.89 DRD4 (0.51) DRD2DRD4DRD3HTR1AHTR7
Bromide SCHEMBL7773422 0.88 DRD4 (0.50) DRD2DRD4DRD3HTR1AHTR7
Bromide SCHEMBL7775356 0.88 OGA (0.41) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL27565727 0.86 NPC1 (0.46) DRD2DRD4DRD3HTR7HTR2A
SCHEMBL7775460 0.85 NPC1 (0.48) DRD2DRD4DRD3HTR7HTR2A
SCHEMBL7773419 0.85 DRD2 (0.61) DRD2DRD4DRD3HTR1AHTR7
Bromide SCHEMBL27545758 0.85 NPC1 (0.46) DRD2DRD4DRD3HTR7HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117663-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2001-07-25 EP disclosed
WO-2000018767-A2 2-PIPERAZINO ALKYLAMINO BENZOAZOLE DERIVATIVES: DOPAMINE RECEPTOR SUBTYPE SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 2000-04-06 WO disclosed