SCHEMBL7775457

SCHEMBL7775457

CC(C)OC(=O)C(C)C#N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
ALDH1A1 P00352 4/20 0.33
MAPT P10636 4/20 0.33
KDM4E B2RXH2 3/20 0.33
HIF1A Q16665 2/20 0.33
MAPK1 P28482 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
CSNK1A1 P48729 1/20 0.32
MEN1 O00255 1/20 0.31
GLA P06280 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
LMNA P02545 4/20 0.30
RAB9A P51151 1/20 0.30
CA12 O43570 3/20 0.30
CA1 P00915 3/20 0.30
CA2 P00918 3/20 0.30
CA7 P43166 3/20 0.30
CA9 Q16790 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718636 0.83 TSHR (0.30) TSHR
SCHEMBL11566231 0.81 DPP4 (0.33)
SCHEMBL11442409 0.80 TSHR (0.42) TSHRALDH1A1MAPTKDM4EHIF1A
SCHEMBL27810375 0.80 TSHR (0.42) TSHRALDH1A1MAPTKDM4EHIF1A
SCHEMBL7645726 0.77
SCHEMBL7436520 0.76 TSHR (0.39) TSHRALDH1A1MAPTKDM4EHIF1A
SCHEMBL9347901 0.75
SCHEMBL18643740 0.75
SCHEMBL28446509 0.75
SCHEMBL2911451 0.75 TSHR (0.42) TSHRHCAR2LMNACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114763319-B Method for co-producing valproamide and sodium valproate 湖南大学 2023-03-31 CN disclosed
US-20170028099-A1 METHOD FOR THE PRODUCTION OF POLY(2-OCTYL CYANOACRYLATE)-POLYISOBUTYLENE CO-NETWORK, AND SUPER INITIATORS THEREFOR THE UNIVERSITY OF AKRON (US) 2017-02-02 US disclosed
WO-2015018797-A2 ANTIVIRAL COMPOUNDS HAPLOGEN GMBH (AT) 2015-02-12 WO disclosed
EP-0839818-B1 Optically active diphosphines, transition metal complex containing the same, and process for producing an optically active compound using the complex TAKASAGO PERFUMERY CO LTD (JP) 2001-08-16 EP disclosed
US-5789609-A CATALYST FOR ASSYMETRIC SYNTHESIS, REACTION OF AN A-CYANO ESTER AND A VINYL KETONE TO PRODUCE AN OXO CYANO ESTER TAKASAGO INTERNATIONAL CORPORATION (JP) 1998-08-04 US disclosed
EP-0839818-A1 Optically active diphosphine, transition metal complex containing the same, and process for producing optically active compound using the complex Takasago International Corporation (JP) 1998-05-06 EP disclosed
US-RE30420-E DIURETIC, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DE) 1980-10-21 US disclosed
US-4112227-A DIURETIC, SALURETIC, ANTIHYPERTENSIVE, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (DE) 1978-09-05 US disclosed
US-4081596-A DIURETIC, SALURETIC, ANTIHYPERTENSIVE, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (DT) 1978-03-28 US disclosed
US-4056533-A HYPOTENSIVE AGENTS, ANTICOAGULANTS, DIURETICS BAYER AKTIENGESELLSCHAFT (DT) 1977-11-01 US disclosed
US-4005215-A DIURETIC BAYER AKTIENGESELLSCHAFT (DT) 1977-01-25 US disclosed
US-4000294-A DIURESIS OR SALURESIS BAYER AKTIENGESELLSCHAFT (DT) 1976-12-28 US disclosed
US-3992404-A DIURETICS, SALURETICS, ANTIHYPERTENSIVE AGENTS, AND ANTITHROMBOTIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-11-16 US disclosed
US-3978077-A DIURETIC, HYPOTENSIVE, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (GB) 1976-08-31 US disclosed
US-3957814-A DIURETICS, SALURETICS, HYPOTENSIVE AGENTS, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (DT) 1976-05-18 US disclosed
US-3952008-A DIURETIC, SALURETIC, HYPOTENSIVE, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed