SCHEMBL7779340

SCHEMBL7779340

CCc1nn(CC(CN)OC(=O)/C=C/C(=O)OC(CN)Cn2nc(CC)c3ccc(C(F)(F)F)cc32)c2cc(C(F)(F)F)ccc12

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 7/20 0.36
PTGDR2 Q9Y5Y4 6/20 0.33
PTGER1 P34995 1/20 0.33
AKR1B1 P15121 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CRHR1 P34998 1/20 0.32
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7776530 0.87 SLC22A12 (0.37) SLC22A12PTGDR2
SCHEMBL7776527 0.86 SLC22A12 (0.38) SLC22A12PTGDR2AKR1B1
SCHEMBL7777106 0.85 SLC22A12 (0.37) SLC22A12
Fumaric Acid SCHEMBL5678111 0.79 SLC22A12 (0.43) SLC22A12PTGDR2PTGER1AKR1B1NPSR1
Fumaric Acid SCHEMBL5678122 0.79 SLC22A12 (0.43) SLC22A12PTGDR2PTGER1AKR1B1NPSR1
SCHEMBL5678114 0.77 DPP7 (0.34) SLC22A12PTGDR2PTGER1AKR1B1NPSR1
SCHEMBL905944 0.76 HTR2A (0.48) SLC22A12
Fumaric Acid SCHEMBL5678117 0.73 SLC22A12 (0.45) SLC22A12PTGDR2PTGER1AKR1B1
SCHEMBL5679817 0.72 PPARG (0.36) SLC22A12PTGDR2CRHR1
SCHEMBL5679829 0.72 PPARG (0.36) SLC22A12PTGDR2CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129078-A2 INDAZOLE DERIVATIVES WITH 5-HT2 RECEPTOR ACTIVITY VERNALIS RESEARCH LIMITED (GB) 2001-09-05 EP disclosed
WO-2000012481-A2 INDAZOLE DERIVATIVES WITH 5-HT2 RECEPTOR ACTIVITY________________ VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed