SCHEMBL7779774

SCHEMBL7779774

CCc1cccc([N+](=O)[O-])c1CC

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.52
TSHR P16473 4/20 0.50
ALDH1A1 P00352 4/20 0.50
FBP1 P09467 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
GPR35 Q9HC97 2/20 0.47
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
S100A4 P26447 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8361517 0.90 TDP1 (0.58) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL14388905 0.89 TDP1 (0.46) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL9077656 0.89 FBP1 (0.50) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL14388907 0.87 TDP1 (0.47) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL18816139 0.87 TSHR (0.59) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL18816130 0.87 TDP1 (0.47) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL9077669 0.86 TDP1 (0.43) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL8730292 0.86 TDP1 (0.43) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL8172704 0.84 FBP1 (0.49) TDP1TSHRALDH1A1FBP1SMN1; SMN2
SCHEMBL18184974 0.84 TDP1 (0.48) TDP1TSHRALDH1A1FBP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9815768-B2 Method for producing 2-(halogenomethyl)-3-methylnitrobenzene SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2017-11-14 US disclosed
US-20160332956-A1 METHOD FOR PRODUCING 2-(HALOGENOMETHYL)-3-METHYLNITROBENZENE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2016-11-17 US disclosed
US-6251903-B1 Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonist COCENSYS, INC. 2001-06-26 US disclosed
EP-1053990-A2 A method of producing an aromatic ketone and an aromatic ketone composition containing it TORAY INDUSTRIES, INC. (JP) 2000-11-22 EP disclosed
US-6147075-A ANALGESICS; PSYCHOLOGICAL DISORDERS COCENSYS, INC. (US) 2000-11-14 US disclosed
EP-0732942-A4 ALKYL, AZIDO, ALKOXY, AND FLUORO-SUBSTITUTED AND FUSED QUINOXALINEDIONES AND THE USE THEREOF AS GLYCINE RECEPTOR ANTAGONISTS COCENSYS INC (US) 2000-03-22 EP disclosed
US-5977107-A Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones and the use thereof as glycine receptor antagonists COCENSYS, INC. (US) 1999-11-02 US disclosed
US-5631373-A NERVOUS SYSTEM DISORDERS STATE OF OREGON, ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION, ACTING FOR AND ON BEHALF OF THE OREGON HEALTH SCIENCES UNIVERSITY AND THE UNIVERSITY OF OREGON, EUGENE OREGON (US) 1997-05-20 US disclosed
EP-0732942-A1 ALKYL, AZIDO, ALKOXY, AND FLUORO-SUBSTITUTED AND FUSED QUINOXALINEDIONES AND THE USE THEREOF AS GLYCINE RECEPTOR ANTAGONISTS ACEA PHARMACEUTICALS, INC. (US) 1996-09-25 EP disclosed
WO-1995012417-A1 ALKYL, AZIDO, ALKOXY, AND FLUORO-SUBSTITUTED AND FUSED QUINOXALINEDIONES AND THE USE THEREOF AS GLYCINE RECEPTOR ANTAGONISTS ACEA PHARMACEUTICALS, INC. (US) 1995-05-11 WO disclosed
US-4502995-A Nucleophilic substitution process ETHYL CORPORATION (US) 1985-03-05 US disclosed
US-4171425-A ANIONIC CATALYST, 2-PYRROLIDONE OR E-CAPROLACTAM CHEVRON RESEARCH COMPANY (US) 1979-10-16 US disclosed
US-4051187-A CARBON CATALYST WITH SYNERGISTIC QUANTITIES OF THODIUM, TRICHLORIDE OR RHODIUM TRIBROMIDE OXAMINE, INC. (US) 1977-09-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160332956-A1 METHOD FOR PRODUCING 2-(HALOGENOMETHYL)-3-METHYLNITROBENZENE CYP1B1, DNMT1, DNMT3A TDP1 2652/4885TSHR 1157/4885ALDH1A1 798/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.