Methylhomatropine

Methylhomatropine

SCHEMBL77827

C[N+]1(C)C2CCC1CC(OC(=O)C(O)c1ccccc1)C2.[Br-]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Methylhomatropine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 5/20 0.97
CHRM1 known ✓ P11229 4/20 0.97
CHRM3 known ✓ P20309 4/20 0.71
CHRM4 known ✓ P08173 3/20 0.62
CHRM5 known ✓ P08912 3/20 0.62
PABPC1 P11940 2/20 0.74
BLM P54132 2/20 0.71
LMNA P02545 2/20 0.64
CYP2D6 P10635 2/20 0.64
CYP2C9 P11712 1/20 0.64
HSD17B10 Q99714 1/20 0.64
APOBEC3A P31941 1/20 0.63
APOBEC3G Q9HC16 1/20 0.63
SMN1; SMN2 Q16637 3/20 0.62
TDP1 Q9NUW8 1/20 0.62
CYP2C19 P33261 1/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
TSHR P16473 1/20 0.55
NR1I2 O75469 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylhomatropine SCHEMBL29555824 1.00 CHRM2 (0.97) CHRM2CHRM1PABPC1CHRM3BLM
Methylhomatropine SCHEMBL20659943 1.00 CHRM2 (0.97) CHRM2CHRM1PABPC1CHRM3BLM
Methylhomatropine SCHEMBL613580 1.00 CHRM2 (0.97) CHRM2CHRM1PABPC1CHRM3BLM
Methylhomatropine SCHEMBL17179980 0.99 CHRM2 (1.00) CHRM2CHRM1PABPC1CHRM3BLM
Methylhomatropine SCHEMBL30516140 0.99 CHRM2 (1.00) CHRM2CHRM1PABPC1CHRM3BLM
Methylhomatropine SCHEMBL16784195 0.99 CHRM2 (1.00) CHRM2CHRM1PABPC1CHRM3BLM
Methylatropine SCHEMBL1321572 0.83 BLM (1.00) CHRM2CHRM1PABPC1CHRM3BLM
Methylatropine SCHEMBL30647266 0.83 BLM (1.00) CHRM2CHRM1PABPC1CHRM3BLM
Phenactropinium SCHEMBL29387827 0.82 CHRM2 (0.70) CHRM2CHRM1PABPC1CHRM3BLM
Phenactropinium SCHEMBL8916468 0.82 CHRM2 (0.70) CHRM2CHRM1PABPC1CHRM3BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1072 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115028628-B RSV-F protein small molecule inhibitor and application thereof in preparation of medicines for preventing and treating RSV infection 中南大学 2023-10-10 CN claimed
EP-4178948-A2 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF Universidade de Santiago de Compostela (ES) 2023-05-17 EP claimed
EP-4154879-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NICOTINE WITHDRAWAL SYMPTOMS Korea Institute of Science and Technology (KR) 2023-03-29 EP claimed
WO-2022023496-A2 FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF UNIVERSIDADE DE SANTIAGO DE COMPOSTELA (ES) 2022-02-03 WO claimed
US-20200397702-A1 PHARMACEUTICAL COMPOSITIONS SHIN NIPPON BIOMEDICAL LABORATORIES, LTD. (JP) 2020-12-24 US claimed
EP-3493789-A2 INTRANASAL PHARMACEUTICAL POWDER COMPOSITIONS Shin Nippon Biomedical Laboratories, Ltd. (JP) 2019-06-12 EP claimed
US-10149822-B2 Compositions and methods for combination ingredient delivery THE FIX, LLC (US) 2018-12-11 US claimed
US-10123996-B2 Macrocyclic lactone compounds and methods for their use ELIXIR MEDICAL CORPORATION (US) 2018-11-13 US claimed
WO-2018025089-A2 PHARMACEUTICAL COMPOSITIONS SHIN NIPPON BIOMEDICAL LABORATORIES, LTD. (JP) 2018-02-08 WO claimed
CN-106432221-B A kind of process for purification of Homatropine Methylbromide 湖北百科亨迪药业有限公司 2018-01-12 CN claimed
WO-2006058249-A9 METHODS AND COMPOSITIONS FOR DETERRING ABUSE OF ORALLY ADMINISTERED PHARMACEUTICAL PRODUCTS ACURA PHARMACEUTICALS INC (US) 2006-07-20 WO claimed
WO-2006058249-A2 METHODS AND COMPOSITIONS FOR DETERRING ABUSE OF ORALLY ADMINISTERED PHARMACEUTICAL PRODUCTS ACURA PHARMACEUTICALS, INC. (US) 2006-06-01 WO claimed
US-20060110327-A1 Methods and compositions for deterring abuse of orally administered pharmaceutical products ACURA PHARMACEUTICALS, INC. 2006-05-25 US claimed
EP-1480677-A2 COMPOSITION FOR STABILIZING HYALURONIC ACID IOLTECH (FR) 2004-12-01 EP claimed
US-20030133986-A1 Compositions for stabilizing poly (carboxylic acids) TSAO FU-PAO (US) 2003-07-17 US claimed
WO-2003043660-A2 COMPOSITION FOR STABILIZING HYALURONIC ACID NOVARTIS AG (CH) 2003-05-30 WO claimed
EP-1233761-A1 OSMOTIC DOSAGE FORM COMPRISING FIRST AND SECOND COATS ALZA Corporation (US) 2002-08-28 EP claimed
WO-2001037815-A1 OSMOTIC DOSAGE FORM COMPRISING FIRST AND SECOND ALZA CORPORATION (US) 2001-05-31 WO claimed
US-5008111-A Pretreating skin with anticholinergic quaternary ammonium salt to suppress perspiration SCHERING CORPORATION (US) 1991-04-16 US claimed
US-4824676-A ANTICHOLINERGIC AGENT TO SUPPRESS PERSPIRATION SCHERING CORPORATION (US) 1989-04-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10123996-B2 Macrocyclic lactone compounds and methods for their use CHRM2, CHRM1, CHRM5 CHRM2 1/4885CHRM1 2/4885CHRM3 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.